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N-cycloheptyl-1-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[1-(pyridin-3-yl)pentyl]acetamide
1-[5-({[2-(3-fluorophenyl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
2-(3-methoxypropyl)-8-[(1R,2R)-2-phenylcyclopropanecarbonyl]-2,8-diazaspiro[4.5]decan-3-one
N-[3-(2-methoxybenzamido)phenyl]-2-methyloxane-2-carboxamide
1-(furan-2-carbonyl)-4-(6-hydroxypyrimidin-4-yl)-1,4-diazepan-6-ol
1,3-dimethyl-6-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
N-[(2R)-1-hydroxy-3-methylbutan-2-yl]-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
N-[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
N-(4-chloro-2-fluorophenyl)-2-[(2-methanesulfonamidoethyl)amino]acetamide
1-(2-benzyl-1,3-thiazole-4-carbonyl)azocane
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-[2-(thiophen-2-yl)ethyl]acetamide
4-[2-(piperidine-1-carbonyl)phenoxy]-1-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidine
4-(benzyloxy)-1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}piperidine
1-(2,3-dihydro-1H-indol-1-yl)-2-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}ethane-1,2-dione
N-[2-(4-fluorophenyl)ethyl]-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetamide
5-{5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}-N,N-dimethylpyrimidin-2-amine
3-(1-butyl-1H-imidazol-2-yl)-1-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
N-cyclopropyl-3-[1-(3,5-dimethylbenzoyl)piperidin-4-yl]propanamide
{4-[(2-chlorophenyl)methyl]piperidin-4-yl}methanol
(3S,4S)-4-(3-methoxyphenyl)-1-[(1-methyl-1H-indol-3-yl)methyl]piperidin-3-ol
4-(4-methanesulfonylphenyl)-2-(methylsulfanyl)pyrimidine
(3R,4R)-4-(azepan-1-yl)-1-{[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}piperidin-3-ol
2-(6,8-dimethyl-4-oxo-3,4-dihydroquinazolin-3-yl)-4-methylpentanamide
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(4-methylphenyl)quinoline-4-carboxamide
1-(2-ethylphenyl)-4-[1-(propan-2-yl)piperidine-4-carbonyl]piperazine
4-(4-{[(3aS,6aS)-3a-(hydroxymethyl)-octahydrocyclopenta[c]pyrrol-2-yl]methyl}phenyl)-2-methylbutan-2-ol
{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}(methyl){[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}amine
(3R,4S)-4-cyclopropyl-1-(4,5-dimethylthiophene-2-carbonyl)-N,N-dimethylpyrrolidin-3-amine
4-{1-[4-(2H-1,3-benzodioxol-5-yl)phenyl]ethyl}morpholine
6-(1,2,3,4-tetrahydroisoquinolin-5-yl)pyridin-3-ol
(3R,5S)-N-[2-(1H-imidazol-4-yl)ethyl]-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
1-[(1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methyl]pyrrolidin-2-one
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propan-1-one
(3S,4R)-1-(8-fluoroquinoline-2-carbonyl)-N,N-dimethyl-4-propylpyrrolidin-3-amine
4-[1-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperidin-4-yl]thiomorpholine
methyl({4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-[4-(2-ethylbutyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[(2E)-3-(pyridin-4-yl)prop-2-enoyl]piperidin-4-yl}propanamide
4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-pyrazole-3-carbonyl)piperidine
N-(1-butyl-1H-pyrazol-5-yl)-2-[3-(dimethyl-1,2-oxazol-4-yl)-1H-indazol-1-yl]acetamide
N-[(4-methyloxan-4-yl)methyl]-2-oxo-2-phenylacetamide
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[2-(2,5-dimethylphenyl)ethyl]acetamide
10-methoxy-5-{2-methylpyrido[2,3-d]pyrimidin-4-yl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
2-(dimethyl-1,2-oxazol-4-yl)-6-methylpyridine-3-carboxamide
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
N,N-dimethyl-4-{5-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-4-phenyl-1H-imidazol-1-yl}butanamide
{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}[1-(thiophen-2-yl)ethyl]amine
1-[1-(5-hydroxypyridine-2-carbonyl)piperidin-3-yl]pyrrolidin-2-one