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8-(butan-2-yl)-3-[2-(dimethylamino)ethyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyrimidin-4-ylmethyl)acetamide
N-(2-methoxyethyl)-4-{[2-(4-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-methyl-2-phenyl-N-(1H-pyrazol-3-ylmethyl)acetamide
3-(benzylsulfanyl)-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]propan-1-one
5-ethyl-N4-[3-(pyridin-3-yloxy)propyl]pyrimidine-2,4-diamine
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-propylpyrimidine-5-carboxamide
1-[(1S)-2,3-dihydro-1H-inden-1-yl]-2-(2,3-dimethoxyphenyl)-1H-imidazole
N-[(4-methoxyphenyl)methyl]-2-methyl-N-(oxolan-2-ylmethyl)-1-benzofuran-5-carboxamide
4-[2-(2-fluorophenyl)ethyl]-3-(1H-indol-3-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4R)-1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
2-(2-methyl-1,3-thiazol-4-yl)-N-(oxolan-2-ylmethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
4-{1-[2-(azepan-1-yl)-2-oxoethyl]pyrrolidin-3-yl}benzoic acid
1-(2-chloroprop-2-en-1-yl)-3-{[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]methyl}-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
1-{2-methyl-2,7-diazaspiro[4.5]decan-7-yl}-4-(1H-pyrazol-4-yl)butan-1-one
2-(4,5-dichloro-1H-imidazol-1-yl)-N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
2,3-dimethyl-6-(2-phenylazetidine-1-carbonyl)quinoxaline
1-[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]-4-phenylpiperidine-4-carbonitrile
3-[(3R,4S)-1-(1H-indol-5-ylmethyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
2-amino-4-[1-(pyridin-3-yl)-1H-pyrrol-2-yl]-6-(trimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
2-acetyl-N-(1-phenylethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-6-ethyl-2-methylquinoline-4-carboxamide
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-hydroxypyridine-2-carboxamide
3-[1-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
N-[2-(2-methylpropanesulfonyl)ethyl]-3-(piperidin-3-yl)benzamide
(1R,5R)-N-(4-fluorophenyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}propanamide
4-[(2-methoxyphenyl)methyl]-3-[2-(morpholin-4-yl)-2-oxoethyl]piperazin-2-one
3-(1H-pyrazol-1-yl)-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N-(cyclopropylmethyl)-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
3,3-dimethyl-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
(1S,4S)-5-(2-fluorobenzoyl)-2-(2-methoxy-5-methylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
1-[cyclopropyl(1-methyl-1H-1,2,4-triazol-5-yl)methyl]-3-{1-[(2-methoxyphenyl)methyl]-1H-pyrazol-5-yl}urea
7-[(4-fluorophenyl)methyl]-2-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
2-[(2-{[(3-propyl-1,2-oxazol-5-yl)methyl]carbamoyl}phenyl)amino]acetic acid
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}azetidine-2-carboxylic acid
3-({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}sulfamoyl)-N-(2-methylpropyl)benzamide
3-(3-hydroxyquinoxalin-2-yl)-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]propanamide
(1R,9aR)-1-{[cyclopropyl(3-phenylprop-2-yn-1-yl)amino]methyl}-octahydro-1H-quinolizin-1-ol
9-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
14-[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-5-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
(3S,4S)-1-[(4-chloro-2-fluorophenyl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
6-[4-(3-chlorophenyl)-2-methyl-5-oxopiperazine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
N-[(3R,4S)-1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
1'-(8-methoxyquinolin-2-yl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
(2S)-2-(2,3-difluorophenyl)-2-[(6-methoxy-3-methyl-1-benzofuran-2-yl)formamido]acetic acid
3-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-1-[3-(1H-1,2,4-triazol-1-yl)phenyl]urea
5-(3-fluorophenyl)-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-1,2,4-triazin-3-amine
N-benzyl-5-{2,8-diazaspiro[4.5]decan-2-ylmethyl}pyrimidin-2-amine
(2S,4S)-4-{[(2,5-difluorophenyl)methyl]amino}-N-ethyl-1-(propan-2-yl)pyrrolidine-2-carboxamide