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N-[3-(dimethylcarbamoyl)-4-methoxyphenyl]-4-(pyrimidin-2-yl)piperazine-1-carboxamide
2-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
4-(1H-imidazol-2-yl)-1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(2,2,2-trifluoroethyl)piperidine-3-carboxamide
4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-2-methylquinoline
N-methyl-1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-(2-phenylethyl)piperidine-4-carboxamide
5-(2-{2-[(dimethylsulfamoyl)amino]ethyl}morpholin-4-yl)-2-methyl-2,3-dihydropyridazin-3-one
N,1-dimethyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[2-methoxy-5-(methylcarbamoyl)phenyl]-3-(pyrrolidin-1-yl)pyrrolidine-1-carboxamide
1-[3-({[3-(4-methyl-1,3-thiazol-5-yl)propyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
2-{4-[2-(2-aminoethyl)quinazolin-4-yl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
4-{3-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]propoxy}benzamide
4-(1-ethyl-1H-imidazol-2-yl)-N-[2-(trifluoromethyl)phenyl]piperidine-1-carboxamide
6-fluoro-3-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]quinolin-4-ol
2-{4-[(4,5-dimethylthiophen-2-yl)methyl]piperazin-1-yl}-5-methyl-1,3-benzoxazole
4-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-tert-butylpyrrolidin-2-one
4-(hydroxymethyl)-4-[(3-methoxyphenyl)methyl]-N,N-dimethylpiperidine-1-sulfonamide
5-hydroxy-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]pyrazine-2-carboxamide
N-(2-methanesulfonylethyl)-3-{[4-(methylamino)piperidin-1-yl]sulfonyl}benzamide
3-{1-[(2-ethylpyrimidin-4-yl)methyl]piperidin-2-yl}propanoic acid
5-(2-{2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}-1H-imidazol-1-yl)-2-methylpyridine
N3-cycloheptyl-1-cyclopropyl-N5-(1-methoxybutan-2-yl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-ethyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-N-[2-(pyridin-2-yl)ethyl]piperidin-4-amine
4-(3-chlorophenoxy)-1-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]piperidine
2-(2-hydroxyethyl)-N-[2-(2-methylphenyl)-1,3-benzoxazol-6-yl]pyrrolidine-1-carboxamide
1-(4-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
4-{1-[1-(4-propyl-1,2,3-thiadiazole-5-carbonyl)piperidin-4-yl]ethyl}morpholine
(3S,4R)-4-(3-fluorophenyl)-1-[4-(1,3-oxazol-5-yl)benzoyl]pyrrolidine-3-carboxylic acid
3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-(pyridin-3-ylmethyl)piperidin-3-yl]-1-(4-methylpiperidin-1-yl)propan-1-one
3-(2-methoxyphenyl)-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}propanamide
2-{1-[3-(dimethylsulfamoyl)propyl]pyrrolidin-3-yl}benzoic acid
dimethyl(3-{2-[1-(4-methylquinolin-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
N-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-N-methyl-1,2,3,4-tetrahydronaphthalen-1-amine
4-(3-fluorophenoxy)-1-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]piperidine-4-carboxylic acid
4-(2-{1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-2-yl}ethyl)phenol
1-{[2-(2,4-dichlorophenoxy)acetamido]methyl}cyclopentane-1-carboxylic acid
3-chloro-6-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]pyridine-2-carboxylic acid
6-methyl-3-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-4-(trifluoromethyl)benzamide
2-{4-[(2-chloro-4,5-dimethoxyphenyl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
4-[(1-acetylpiperidin-4-yl)oxy]-3-chloro-N-[2-(dimethylamino)ethyl]benzamide
8-[(3E)-hex-3-enoyl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(6-methoxy-2H-chromen-3-yl)methyl]-4-(2-methylpyridin-4-yl)piperazine
2-(1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-imidazol-2-yl)pyridine
[1-(3-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}phenyl)ethyl]dimethylamine
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-pyrrole-2-carboxamide
dimethyl(2-{[(3-methylthiophen-2-yl)methyl]({[6-(trifluoromethyl)pyridin-3-yl]methyl})amino}ethyl)amine
(4aS,7aR)-1-[(3-chloro-4,5-dimethoxyphenyl)methyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(3-methylpyridin-2-yl)methyl]-4-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)piperazine
2-{1-[(dimethyl-1,3-thiazol-5-yl)methyl]-1H-imidazol-2-yl}-5-ethylpyridine