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1-(3-methyl-5-{5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-yl}-1H-1,2,4-triazol-1-yl)butan-2-ol
[1-(furan-2-yl)ethyl](methyl)({2-[3-(4-methylpiperazin-1-yl)propoxy]phenyl}methyl)amine
1-{[2-(2-fluoro-3-methoxyphenyl)-1H-imidazol-1-yl]methyl}cyclohexan-1-ol
1-[(4-fluoro-3-methoxyphenyl)methyl]-3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
N-butyl-5-methyl-4-{methyl[2-(pyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
5-(methanesulfonylmethyl)-2-[2-(trifluoromethoxy)phenyl]pyridine
ethyl 4-[5-cyclohexaneamido-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carbonyl]piperazine-1-carboxylate
[(3R,4R)-1-({2,4-dimethyl-5-[(4-methylpiperidin-1-yl)methyl]phenyl}methyl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
8-[2-(morpholin-4-yl)acetyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
(4aS,8aS)-4a-hydroxy-N-(2-methoxy-5-methylphenyl)-decahydroisoquinoline-2-carboxamide
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}propanamide
7-(2-hydroxyethyl)-2-[1-(1H-imidazol-1-ylmethyl)cyclopropanecarbonyl]-2,7-diazaspiro[4.5]decan-6-one
N-propyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-cyclopropyl-3-[1-(3-phenylprop-2-ynoyl)piperidin-4-yl]propanamide
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(2-hydroxy-3-methoxypropyl)amine
N-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-(pyrimidin-2-yl)piperidin-3-amine
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-2-(4-fluorophenyl)azetidine
2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)acetamide
5-(benzylamino)-1-(cyclohexylmethyl)-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
6-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1,3-benzothiazole
2-({3-[(4-phenylbutan-2-yl)carbamoyl]phenyl}amino)acetic acid
2-cyclopropanecarbonyl-8-(6-methylpyridazin-3-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
2-(3-methyl-1,2-oxazol-5-yl)-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]acetamide
ethyl 4-[9-methoxy-7-(6-methoxypyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidine-1-carboxylate
6-{2-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1H-imidazol-1-yl}quinoxaline
2-{2-[6-(dimethylcarbamoyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-3-yl]acetamido}acetic acid
2-[4-(adamantan-1-yl)piperazine-1-carbonyl]pyrazine
[(3R,4S)-4-[(4-methylpiperazin-1-yl)methyl]-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]methanol
(3S,4R)-4-(2-methoxyphenyl)-1-[2-oxo-2-(piperidin-1-yl)ethyl]pyrrolidine-3-carboxylic acid
(2E)-1-{4-[5-(3-fluorophenyl)-2-[(2-methoxyethyl)sulfanyl]pyrimidin-4-yl]piperidin-1-yl}-3-(1H-imidazol-4-yl)prop-2-en-1-one
1-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
N-{1-[(4-chlorophenyl)methyl]cyclopropyl}-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
8-(3-ethoxypropanoyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-(pyrrolidine-1-sulfonyl)-5-(1H-1,2,3-triazol-1-yl)benzoic acid
(1S,4S)-2-[2-(methylsulfanyl)phenyl]-5-[(5-methylthiophen-2-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
5-{[5-(3-methyl-1-benzofuran-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1H-1,2,3,4-tetrazole
4-{2-[2-(4-methoxyphenyl)-1H-imidazol-1-yl]ethyl}benzene-1-sulfonamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-phenoxyacetamide
1-[2-(morpholin-4-ylmethyl)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[2-(2,6-dimethylmorpholin-4-yl)ethyl]-2,4-dimethyl-1,3-thiazole-5-carboxamide
1'-[(5-ethylpyridin-2-yl)methyl]-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-[1-(furan-2-ylmethyl)piperidin-4-yl]pyrimidin-4-amine
[(5-tert-butyl-1H-pyrazol-3-yl)methyl](methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
(1R,5S,6S)-6-(morpholine-4-carbonyl)-3-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
methyl 1-[(3S,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-(furan-3-ylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-[(4-ethylphenyl)methyl]-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
3,4-difluoro-N-({3-methoxy-4-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzene-1-sulfonamide