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N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-4-fluorobenzene-1-sulfonamide
[(2-methoxyphenyl)methyl][3-(methylsulfanyl)propyl](prop-2-en-1-yl)amine
2-[(3R,4S)-3-[(dimethylsulfamoyl)amino]-4-propylpyrrolidin-1-yl]-N-ethylpyrimidin-4-amine
(3R,4R)-1-{[3-(4-chlorophenoxy)phenyl]methyl}-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
3-cyclopropyl-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
7-(4-chlorophenyl)-2-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
methyl 2-[({1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}carbamoyl)amino]benzoate
3-cyclohexyl-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
4-acetamido-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}butanamide
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(4-fluoro-2-methylphenyl)ethan-1-one
1-[(2-fluorophenyl)methyl]-6-oxo-N-[3-(pyridin-3-yl)propyl]piperidine-3-carboxamide
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclohex-3-ene-1-carboxamide
5-{[5-(2-chlorophenyl)furan-2-yl]methyl}-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(furan-3-ylmethyl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
(1R,5S)-N-(1H-indazol-7-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]oxolane-3-carboxamide
2-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-(1-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazole
N,4-dimethyl-N-{2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}-1,2,5-oxadiazole-3-carboxamide
2-[1-(1-propylpiperidin-4-yl)-1H-imidazol-2-yl]quinoline
4-{[1-ethyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methyl}morpholine
8-(2-methoxyacetyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-hydroxyethan-1-one
ethyl 2-[1-(2-{2,5-dioxo-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidin-3-yl}acetyl)piperidin-2-yl]acetate
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-fluoro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-1,3-dimethyl-1H-pyrazole-5-carboxamide
1-ethyl-3-(4-methylpiperazine-1-carbonyl)-N-(2,2,2-trifluoroethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{[2-(2H-1,3-benzodioxol-5-yl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenol
N-(1-oxo-1,3-dihydro-2-benzofuran-5-yl)-2-[2-(thiophen-2-yl)ethyl]piperidine-1-carboxamide
6-ethyl-2-methoxy-3-{[(4-methylpyrimidin-2-yl)amino]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]urea
1-(butan-2-yl)-5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-N-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
3-(1H-imidazol-2-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}benzamide
4-(hydroxymethyl)-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]azepan-4-ol
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-1,3-oxazole-4-carboxamide
1-(2-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
1-{4-[2-(4-fluorophenyl)piperidine-1-carbonyl]phenyl}ethan-1-one
3-({5-[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}methyl)pyridine
2-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-2-[4-(methylsulfanyl)phenyl]acetic acid
4-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-1-[(3-fluorophenyl)methyl]piperazin-2-one
({5-[4-(azepan-1-ylmethyl)phenyl]-1,2,4-oxadiazol-3-yl}methyl)dimethylamine
N,2,3-trimethyl-N-[(1,2,2-trimethylpyrrolidin-3-yl)methyl]-1H-indole-7-carboxamide
N-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-2-(4,5-dichloro-2-methyl-1H-imidazol-1-yl)acetamide
2-(carbamoylmethyl)-N-[3-(3-methoxyphenyl)phenyl]piperidine-1-carboxamide
2-amino-6-(1,2-dimethyl-1H-indol-3-yl)-4-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
2-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-6-methylpyridine-3-carbonitrile
6-methyl-N-[(3R,5S)-1-methyl-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-5-phenyl-1,2,4-oxadiazole
N-methyl-2-(piperidin-1-yl)-N-(pyridin-3-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
7-[(4-fluorophenyl)methyl]-2-(furan-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
5-oxo-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide