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2-(2H-1,2,3-benzotriazol-2-yl)-1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-(3-chloro-6-oxo-1,6-dihydropyridazin-1-yl)-N-[2-(dimethylamino)ethyl]-N-[(5-methylthiophen-2-yl)methyl]acetamide
2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyrazin-2-yl)ethyl]acetamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
3-{[(1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-yl)oxy]methyl}pyridine
3-{2-ethyl-3H-imidazo[4,5-b]pyridin-6-yl}-5-[2-(piperidin-2-yl)ethyl]phenol
N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide
3-hydroxy-1-(2-methoxyethyl)-3-{[methyl(quinolin-3-ylmethyl)amino]methyl}piperidin-2-one
N-[1-(furan-2-carbonyl)piperidin-3-yl]-3-azaspiro[5.5]undecan-9-amine
7-cyclohexyl-2-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-7-(1H-inden-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-ethyl-2-oxo-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1,2-dihydropyridine-4-carboxamide
1-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-3-[(dimethylamino)methyl]pyrrolidin-3-ol
4-(2,6-dimethylpyridin-3-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-({1-[(2R)-2-amino-3-(4-chlorophenyl)propanoyl]piperidin-4-yl}methyl)acetamide
9-(3-amino-3-phenylpropanoyl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
3-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidine-1-carbonyl]-1-methyl-1,2-dihydroquinoxalin-2-one
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(phenylamino)pyrimidine-5-carboxamide
N,5,7-trimethyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]pyrido[2,3-d]pyrimidin-4-amine
2-amino-4-(2-methoxypyrimidin-5-yl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-butyl-2-[N-methyl-1-(2-methylfuran-3-yl)formamido]acetamide
N-[3-(azepan-1-yl)propyl]-N-methyl-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
7-{2-[(4-chlorophenyl)sulfanyl]acetyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
{1-[7-(1,2-oxazole-3-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidin-3-yl}methanol
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]pyridine-3-carboxamide
2-[methyl({4-methyl-5-[1-(4-methyl-1H-imidazole-5-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
2-(4-amino-3-methoxypyridin-2-yl)benzamide
1-{1-[(3-methylquinoxalin-2-yl)methyl]piperidin-4-yl}piperidin-3-ol
5-methyl-4-[(pyridin-2-ylmethyl)amino]-N-[1-(thiophen-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
5-amino-N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-1H-pyrazole-3-carboxamide
3-{2-[4-(cyclopropylmethyl)piperazin-1-yl]-2-oxoethyl}-4-[(3,4-difluorophenyl)methyl]piperazin-2-one
2-cyclopropyl-4-{4-[4-(furan-2-carbonyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-({[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}amino)acetamide
1-[(3-fluorophenyl)methyl]-4-[(3-methylthiophen-2-yl)methyl]piperazin-2-one
2-[4-methoxy-2-(1H-pyrazol-1-yl)phenyl]-5-(piperidine-1-carbonyl)pyridine
2-hydroxy-5-({methyl[2-(morpholin-4-yl)propyl]amino}methyl)benzoic acid
N-methyl-N-(1-methylpiperidin-4-yl)-3-{1-[2-(2-oxopiperidin-1-yl)acetyl]piperidin-3-yl}propanamide
(2S,4S)-N-ethyl-4-{[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]amino}-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
4-[(1R)-1-(4-fluorophenyl)ethyl]-3-[(propan-2-yloxy)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[6-oxo-4-(piperazin-1-yl)-1,6-dihydropyridazin-1-yl]-N-propylpropanamide
4-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butanamide
2-{3-butyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-3-(piperidin-1-yl)pyridine
1,6-dimethyl-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(1,3-thiazol-2-yl)-3-{[1-(thiophen-2-yl)propan-2-yl]amino}propanamide
6-methyl-2-(2-methyloxane-2-carbonyl)-5-[5-(1H-pyrrol-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
(1R,7S)-3-tert-butyl-6-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
5-{[4-(3,3-diethylpyrrolidine-1-carbonyl)-1,3-oxazol-2-yl]methoxy}-2-methyl-1,3-benzothiazole
1-[(2-chlorophenyl)methyl]-2-(propan-2-yl)-1H-imidazole