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4-(2-methylpiperidin-1-yl)-3-[3-(4H-1,2,4-triazol-4-yl)benzamido]benzamide
4-[4-(3-methoxypropyl)piperazine-1-carbonyl]-1,2-dihydroisoquinolin-1-one
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[1-(thiophen-3-yl)propan-2-yl]amine
({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
3-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(2-methoxyphenoxy)ethan-1-one
(1S,3R)-3-amino-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}cyclopentane-1-carboxamide
5-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-phenyl-1H-imidazole-4-carboxamide
4-(piperidin-1-yl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}butanamide
1-(1-benzylpiperidine-2-carbonyl)-4-(3-methylpyridin-2-yl)piperazine
(1S,5R)-6-(cyclobutylmethyl)-3-(2,5-dimethylbenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1S,4S)-2-(3-chlorophenyl)-5-(2-methylpropyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
3-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-1-[2-methyl-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]urea
2-{[4-(4-benzyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}benzoic acid
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
1-cyclopentyl-N3-(3-methylbutyl)-4-oxo-N5-[2-(pyridin-3-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-[2-(3-benzyl-1H-1,2,4-triazol-5-yl)ethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{7-[(4-methyl-1,3-thiazol-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}morpholine
4-(4-benzyl-1H-pyrazol-5-yl)-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidine
N-[(3-chlorophenyl)methyl]-2-[4-(2-phenylethyl)morpholin-3-yl]acetamide
4-{2-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-oxoethyl}piperazin-2-one
3-(1H-1,2,3-benzotriazol-5-yl)-1-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]urea
1,3-dimethyl-N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
8-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)thian-4-amine
1-{2-[(3S,4R)-3-cyclopropyl-4-{[ethyl(methyl)sulfamoyl]amino}pyrrolidin-1-yl]ethyl}pyrrolidin-2-one
2-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
N-(3-methylphenyl)-3-({2-oxo-1,3-dioxa-8-azaspiro[4.5]decan-8-yl}methyl)benzamide
5-methyl-5-(4-methylpent-3-en-1-yl)-1-[2-(pyridin-4-yl)ethyl]piperidin-2-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
3-(1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}pyrrolidin-2-yl)-5-methyl-1,2-oxazole
6-({[2-(1H-imidazol-1-yl)phenyl]methyl}amino)pyridine-3-carboxamide
(2R,3R,6R)-5-(5-chloropyridine-2-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(1H-pyrazol-1-yl)-N-{3-[(pyridin-3-yl)amino]propyl}butanamide
[(1-cyclohexylpiperidin-3-yl)methyl][(2-fluorophenyl)methyl](pyridin-3-ylmethyl)amine
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)acetamide
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-N-ethylpiperidine-1-carboxamide
5-{[(5-methanesulfonyl-2-methylpyrimidin-4-yl)amino]methyl}-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
(3aS,6aS)-2-acetyl-5-{[(2-phenylethyl)carbamoyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)(methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-(furan-2-ylmethyl)acetamide
1-(4-ethoxy-3-methylphenyl)-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}butane-1,4-dione
3-[4-(2-methoxybenzoyl)piperazine-1-carbonyl]piperidine-1-carboxamide
N-[(3-methoxyphenyl)methyl]-3-[1-(4,4,4-trifluorobutanoyl)piperidin-3-yl]propanamide
3-ethyl-8-(1H-imidazol-2-ylmethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(3S,4R)-1-[3-(2,4-difluorophenyl)propanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
N,5-dimethyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1-propyl-1H-pyrazole-4-carboxamide
3-[2-oxo-2-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)ethyl]-3,4-dihydroquinazolin-4-one
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propanamide