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N-(2-methoxyethyl)-2-(1-methyl-1H-imidazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-(2,3-dihydro-1H-inden-2-yl)-1-[3-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
[3-(2-methoxyethyl)-1-(5-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]methanol
3-{5-[(2-{[(3S)-3-fluoropyrrolidin-1-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)methyl]thiophen-2-yl}-1H-pyrazole
2-(2-chloro-4-fluorophenoxymethyl)-N-ethyl-N-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide
2-(2,5-dioxoimidazolidin-1-yl)-N-methyl-N-(quinolin-5-ylmethyl)acetamide
1-(oxolane-3-carbonyl)-4-phenyl-1,4-diazepane
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
1-(2H-1,3-benzodioxole-5-carbonyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
2-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-4-methylphenol
2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methoxyphenyl]-5-(methanesulfonylmethyl)pyridine
1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(3-fluorophenoxy)ethan-1-one
2-(dimethylamino)-2-(3-fluorophenyl)-1-{4-[(3-hydroxyphenyl)methyl]piperazin-1-yl}ethan-1-one
8-[(3-chloro-2-fluorophenyl)methyl]-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
(4aR,7aS)-1-{2-[benzyl(methyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(1S,4S)-5-(3-chlorophenyl)-6-oxo-2,5-diazabicyclo[2.2.1]heptan-2-yl]-N-(furan-2-ylmethyl)propanamide
(1R,5R)-N,N-dimethyl-6-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
5-[5-(cyclohex-3-en-1-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
N-[(2-methylphenyl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-ethyl-N-(2-methylprop-2-en-1-yl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
8-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
5-{1-[3-(trifluoromethyl)phenyl]propan-2-yl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
N-butyl-5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-1-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
methyl 2-{4-[(thiolan-3-yl)amino]piperidin-1-yl}acetate
N'-[2-(propan-2-yl)phenyl]-N-[1-(1,3-thiazol-2-yl)propyl]butanediamide
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
5-(morpholin-4-yl)-2-(pyridin-2-ylmethyl)-2,3-dihydropyridazin-3-one
4-{7-[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-5-yl}pyridine
1-[1-(3-cyclopentylpropanoyl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
1-{2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine-3-carbonitrile
1-ethyl-N-[(4-methoxyphenyl)methyl]-5-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[2-(3-methoxyphenyl)-1-{1-[4-(methylsulfanyl)benzoyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
N-[3-(2-methyl-1H-imidazol-1-yl)propyl]-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]propanamide
2-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)pyridin-3-ol
6-(2-phenylethyl)-2-[4-(pyrrolidin-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
2-[2-(dimethylamino)ethyl]-8-(6-methyl-4-oxo-1,4-dihydropyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
[2-(3-ethyl-3-methylpiperidine-1-carbonyl)pyridin-4-yl]methanol
1-(diethylamino)-3-[2-methoxy-4-({[2-(methylsulfanyl)ethyl]amino}methyl)phenoxy]propan-2-ol
(3R,4R)-1-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]-4-ethylpiperidine-3,4-diol
2-[4-(6-ethylpyrimidin-4-yl)piperazine-1-carbonyl]-3,4,7-trimethyl-1H-indole
N-(3-cyclopentylpropyl)-2-(dimethylamino)-2-(2-fluorophenyl)acetamide
3-(3-hydroxyquinoxalin-2-yl)-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]propanamide
2-{1-cyclopentyl-4-[(3,4-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-methyl-5-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1,3-oxazole
3-methyl-6-{5-[1-(pyrrolidin-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}pyridazine
1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(pyridin-3-yl)propan-1-one
2-methyl-N-[4-(pyridin-2-yl)pyrimidin-2-yl]-4,5,6,7-tetrahydro-1,3-benzothiazol-4-amine
3-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyridin-2-ol
4-acetyl-N-[(trimethyl-1H-imidazol-2-yl)methyl]benzamide
3-[4-(1-hydroxy-3-phenylpropyl)piperidine-1-carbonyl]benzene-1,2-diol