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4-ethyl-6-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(pyrrolidine-1-carbonyl)piperidine
4-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-fluoropyridine
3-ethoxy-4-(prop-2-en-1-yloxy)-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]benzamide
6-(1-propyl-1H-1,2,4-triazol-5-yl)quinoline
1-cyclopentanecarbonyl-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
5-[3-(1,3-benzothiazol-2-yl)propanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-[2-(cyclohex-1-en-1-yl)ethyl]-4-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
2-oxo-N-[4-(1,3-thiazol-4-yl)phenyl]-1,3-dioxa-8-azaspiro[4.5]decane-8-carboxamide
2-(3-methoxyphenyl)-5-[1-(1-methoxypropan-2-yl)-1H-imidazol-2-yl]-1,3-thiazole
8-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
(4aR,7aS)-1-methanesulfonyl-4-(pyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N4-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
[2-(1H-imidazol-1-yl)ethyl](methyl){[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
3-(pyridin-2-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-pyrazole-5-carboxamide
2-fluoro-N-({3-methyl-7-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)benzamide
3-(2-chlorophenoxymethyl)-4-(1,3-dimethyl-1H-pyrazol-5-yl)-4H-1,2,4-triazole
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-[(3-methylthiophen-2-yl)methyl]-1,2-oxazole-3-carboxamide
2-[1-(4-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-methylacetamide
methyl 2-{2-[3-oxo-3-(pyrrolidin-1-yl)propyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}acetate
(3R,4R)-1-(1-benzofuran-2-ylmethyl)-4-(morpholin-4-yl)piperidin-3-ol
6-propyl-2-(2-{[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
5-methyl-3-(pyrimidin-5-yl)-1H-indole
1-[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-indol-3-yl)ethan-1-one
3-(2-methoxyethyl)-1-methyl-5-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-1,2,4-triazole
2-[(3,5-difluorophenyl)methyl]-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-(naphthalen-1-ylmethyl)-1,4-diazepan-5-one
4-{2-[2-(2-chloro-6-fluorophenyl)-1H-imidazol-1-yl]ethyl}pyridine
1-(carbamoylmethyl)-N-[2-(quinolin-8-yloxy)ethyl]piperidine-3-carboxamide
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-[3-(dimethylamino)-2-methylpropyl]pyrimidin-2-amine
6-{3-[3-(4-ethylpiperazin-1-yl)propyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}pyridine-3-carbonitrile
ethyl 3-({1-[(2-methoxyphenyl)methyl]-5-[(3-methylbutyl)carbamoyl]-4-oxo-1,4-dihydropyridin-3-yl}formamido)propanoate
2-(4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperazin-1-yl)-1-(piperidin-1-yl)ethan-1-one
3-acetamido-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]propanamide
{4-[(5-ethylpyridin-2-yl)methyl]-1,4-oxazepan-6-yl}methanol
N4-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-N2-cyclopropyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-[2-(3-hydroxypyrrolidin-1-yl)-2-oxoethyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2,3-dihydropyridazin-3-one
4-[(2R)-2-phenylbutyl]thiomorpholine
2-{2-[1-(azepane-1-sulfonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-[4-(4-methylpiperazin-1-yl)pentanoyl]-1-phenylpiperazin-2-one
N,8-dimethyl-3-{[methyl(oxan-4-yl)amino]methyl}-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
(3R,4R)-4-ethyl-1-(2-methyl-1,3-thiazole-5-carbonyl)piperidine-3,4-diol
2-methoxy-1-(1'-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)ethan-1-one
3-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidine-1-carbonyl}-4,5,6,7-tetrahydro-1H-indazole
3-(2-{[2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethyl)-1,3-oxazolidin-2-one
1,3,6-trimethyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1H-pyrazolo[3,4-b]pyridine-4-carboxamide
(3E)-N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}-4-phenylbut-3-enamide
1-(ethanesulfonyl)-4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine