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4-methoxy-2-{[4-(3-methylquinolin-2-yl)piperazin-1-yl]methyl}phenol
1-[(3,4-dimethoxypyridin-2-yl)methyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
methyl 2-(3-methylphenyl)-2-[3-(1,2-oxazinan-2-yl)propanamido]acetate
5-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]thiophene-2-carboxylic acid
N-methyl-N-{1-[1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,2,5,6-tetrahydropyridin-3-yl]propyl}acetamide
2-[4-(2-phenylethyl)-1-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
[(3R,4R)-1-[(2-ethylphenyl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-4-sulfamoylbenzamide
2-{[1-(3-chloro-4-methylphenyl)piperidin-4-yl]amino}-N-ethylpropanamide
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]({[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl})methylamine
(1H-1,3-benzodiazol-2-ylmethyl)(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
N-benzyl-5-[4-(4-chlorophenyl)piperazine-1-carbonyl]-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[(3R,4S)-1-[(3-cyanophenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]oxane-4-carboxamide
1-cyclopentyl-N3,N3-diethyl-4-oxo-N5-{[3-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-2-(1-methyl-1H-pyrrol-3-yl)acetamide
2-hydroxy-1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-4-(methylsulfanyl)butan-1-one
1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-3-propylpiperidine-3-carboxylic acid
4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
(1R,3S)-3-methoxy-3-methyl-7-(pyridin-4-yl)-7-azaspiro[3.5]nonan-1-ol
3-{[3-(2-methyl-1,3-thiazol-4-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
N-[3-(4-fluorophenyl)phenyl]-3-(pyrrolidin-1-yl)pyrrolidine-1-carboxamide
N-benzyl-N,1-dimethyl-5-[(propan-2-yl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-methyl-N-[2-(morpholin-4-yl)ethyl]-1-[4-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-1,3-benzodiazole-5-carbonitrile
6-methyl-2-(pyridin-3-yl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]pyrimidin-4-amine
3-benzoyl-1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)piperidine
4-({1-methyl-2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}carbonyl)benzene-1-sulfonamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-N'-(2-ethoxyphenyl)propanediamide
5-tert-butyl-3-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1H-pyrazole
1-[2-(dimethylamino)ethyl]-5-oxo-N-[2-(pyrazin-2-yl)ethyl]pyrrolidine-3-carboxamide
4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperidine
5-(morpholin-4-ylmethyl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]furan-3-carboxamide
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]propanamide
{[6-(thiophen-3-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}({[2-(trifluoromethyl)phenyl]methyl})amine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-5-(2,6-dimethoxyphenyl)-1,2,4-triazin-3-amine
4-[(2-chloro-4-fluorophenyl)methyl]-3-{2-[4-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
3-[1-(oxolan-3-ylmethyl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
N-(2-methoxyethyl)-3,5-dimethyl-N-(1,3-thiazol-2-ylmethyl)-1-benzofuran-2-carboxamide
(3S,4R)-4-(3-methylthiophen-2-yl)-1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-3-ol
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
1-(4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)pent-4-en-1-one
1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-2-(3-methoxyphenoxy)ethan-1-one
2-amino-6-(3-hydroxyphenyl)-4-[1-(pyridin-4-yl)-1H-pyrrol-2-yl]pyridine-3-carbonitrile
2-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl}quinoxaline
1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-4-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-1,4-diazepane
N-[4-(methylsulfanyl)phenyl]-4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
3,3,3-trifluoro-N-(isoquinolin-5-ylmethyl)-N-methylpropanamide
2-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-6-methylpyridine-3-carboxylic acid
4-(3-hydroxypropanoyl)-1-(2-methylphenyl)piperazin-2-one
N-[2-(dimethylamino)ethyl]-N-[(3-methylthiophen-2-yl)methyl]-3-(pyridin-3-yl)propanamide