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(4aR,7aS)-1-ethyl-4-[2-(2,2,3,3-tetrafluoropropoxy)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{[1-(5-tert-butyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]methyl}pyrrolidin-2-one
5-[4-(3-chlorophenyl)piperazine-1-carbonyl]-1-cyclopentyl-N-methyl-N-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
{[4-(butan-2-yloxy)-3-chlorophenyl]methyl}({5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl})amine
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-(furan-2-yl)-7-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(1S,4S)-2-(3-chlorophenyl)-5-[(2,4,5-trimethoxyphenyl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
9-[(2,3-difluorophenyl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
(3S,4R)-4-(3-methoxyphenyl)-1-[(5-methylfuran-2-yl)methyl]pyrrolidine-3-carboxylic acid
8-(isoquinolin-1-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(7-chloro-2-ethyl-3-methyl-1-benzofuran-5-yl)-2-(morpholin-3-yl)acetamide
N-methyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-(oxan-4-ylmethyl)acetamide
5-[3-(3-methoxypropyl)piperidine-1-carbonyl]-4-methyl-2-(piperidin-1-yl)pyrimidine
1-ethyl-N-(furan-2-ylmethyl)-5-[(3-hydroxy-2,2-dimethylpropyl)amino]-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(dimethyl-1,2-oxazol-4-yl)-3-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)urea
(4aR,7aS)-4-(2,6-dimethylpyrimidine-4-carbonyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
4-(2-methylpiperidin-1-yl)-3-[4-(1H-1,2,4-triazol-1-yl)butanamido]benzamide
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-methanesulfonylpiperidine
2,6,6-trimethyl-3-[2-(4-methyl-3-oxopiperazin-1-yl)-2-oxoethyl]-1-propyl-4,5,6,7-tetrahydro-1H-indol-4-one
3-{[4-(1H-pyrazol-3-yl)piperidin-1-yl]methyl}piperidin-3-ol
1-{2-[methyl(pyridin-2-ylmethyl)amino]acetyl}-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
1-methyl-3-phenyl-8-(3-propyl-1H-pyrazole-4-carbonyl)-1,8-diazaspiro[4.5]decane
(2S,4S)-1-(2-ethoxyacetyl)-N-ethyl-4-(thiophene-2-amido)pyrrolidine-2-carboxamide
5-(4-cyclohexylphenyl)-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1,2,4-triazin-3-amine
3-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1-(2,4,6-triethylphenyl)urea
3-(2-methyl-1H-imidazol-1-yl)-1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
3,5-dimethyl-2-({4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)-1,4-dihydropyridin-4-one
5-(1-cycloheptyl-1H-1,2,3-triazol-4-yl)-3-(2-methoxyethyl)-1,2,4-oxadiazole
2-{5-[pyridin-3-yl(pyrrolidin-1-yl)methyl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
3-[(5-methylfuran-2-yl)methyl]-1-[4-(oxolan-2-ylmethoxy)phenyl]urea
4-{[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]methyl}-N-(trimethyl-1H-pyrazol-4-yl)benzamide
4-{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}morpholine
1-[(4-chlorophenyl)methyl]-5-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-[1-(4-fluorophenyl)-2-methylpropan-2-yl]acetamide
4-ethyl-1-methyl-3-[(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(3R,4R)-4-cyclopropyl-3-methyl-1-(2-propoxybenzoyl)piperidin-4-ol
3-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]-1H-indole
N-[(2,4-difluorophenyl)methyl]-2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
N-[(4-fluorophenyl)methyl]-N-(pyridin-4-ylmethyl)-2-(trimethyl-1H-pyrazol-1-yl)acetamide
N-{[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]methyl}-4-phenylbenzamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
({4-cyclopropyl-5-[1-(oxan-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
2-{1-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-yl}ethan-1-ol
4-({3-[benzyl(methyl)amino]piperidin-1-yl}methyl)-2,6-dimethoxyphenol
N-benzyl-3-{[1-(pyrimidin-5-ylmethyl)piperidin-4-yl]oxy}benzamide
3-acetyl-N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-1H-pyrazole-5-carboxamide
4-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pyridin-2-amine
2-{5-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
2-[5-(oxolan-3-ylmethyl)-1-propyl-1H-1,2,4-triazol-3-yl]acetamide
1-(4-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
3-{[3-(hydroxymethyl)morpholin-4-yl]methyl}-1-methyl-1,2-dihydroquinolin-2-one