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N-(cyclopropylmethyl)-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-propyl-1,3-oxazole-4-carboxamide
4-[4-(difluoromethoxy)benzoyl]-5-methyl-1-(3-methylphenyl)piperazin-2-one
5-[4-(furan-3-carbonyl)-1,4-diazepane-1-carbonyl]-2,3-dimethyl-1H-indole
2-[5-(3,4-dihydro-2H-1-benzopyran-3-yl)-3-[(4-methoxyphenyl)methyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-(furan-2-ylmethyl)-N-methyl-4-oxo-3,4-dihydroquinazoline-2-carboxamide
2-butoxy-1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
N-[(3-methyl-1-benzofuran-2-yl)methyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
1-cyclopentyl-N-(2-{imidazo[1,2-a]pyrimidin-2-yl}ethyl)-6-oxopiperidine-3-carboxamide
1-[2-amino-7-methyl-4-(3-methylphenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
methyl 2-{[(4-chlorophenyl)methyl]sulfamoyl}-6-[(2E)-4-methylpent-2-enoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(4-chloro-1H-pyrazol-1-yl)-1-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propan-1-one
1-(3-{1-oxa-8-azaspiro[4.5]decan-8-yl}-3-oxopropyl)-1,2-dihydropyridin-2-one
3-benzyl-5-(4-methoxy-2-methylphenyl)-1H-1,2,4-triazole
4-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
N-[(3S,4R)-4-(4-methylphenyl)-1-(4-sulfamoylbutanoyl)pyrrolidin-3-yl]acetamide
2-({[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}sulfanyl)pyrimidine
1-(1-{[1-(thiophene-2-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-ol
N-(3-hydroxypropyl)-2-[(3S)-3-hydroxypyrrolidin-1-yl]-N,1-dimethyl-1H-1,3-benzodiazole-5-carboxamide
4-benzyl-3-ethyl-1-[(4-methyl-1H-imidazol-5-yl)methyl]-1,4-diazepan-5-one
2-(2-hydroxyethyl)-9-[2-(methylamino)pyridine-4-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[1-(3,5-dimethylbenzoyl)piperidin-4-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
3-{methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]sulfamoyl}-N-(pyrrolidin-3-yl)benzamide
2-{5-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
3-[(3R,7S,8aS)-3-[(benzylsulfanyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-fluoro-2-methylphenyl)urea
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-N-methyl-4-{[(3-phenoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
2-{2-oxo-8-[6-oxo-1-(propan-2-yl)piperidine-3-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetic acid
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
(benzylsulfamoyl)(pyridin-3-ylmethyl)amine
methyl (2S,4R)-1-methyl-4-{2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetamido}pyrrolidine-2-carboxylate
7-(3-chlorothiophene-2-carbonyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(2S)-N-[4-(3-methoxyphenyl)phenyl]-1-(thiophen-3-ylmethyl)pyrrolidine-2-carboxamide
3-[3-(1-methyl-1H-pyrazol-3-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]propanoic acid
1-{4-[(3S,4S)-3-hydroxy-4-(pyrrolidin-1-yl)pyrrolidin-1-yl]-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
1-{[1-(5-methyl-1,3-benzoxazol-2-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
2-{[(furan-2-ylmethyl)(3-methylbutan-2-yl)amino]methyl}-6-methylpyridin-3-ol
N-(1-cycloheptylpiperidin-3-yl)-3-(1,2-oxazolidin-2-yl)propanamide
methyl 3-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanoate
4-benzyl-3-{1-[6-(dimethylamino)pyrimidin-4-yl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(2R)-2-{[5-(3-fluorophenoxymethyl)-1H-pyrazol-3-yl]formamido}-3-methylbutanamide
1-(furan-3-ylmethyl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
7-[(1-propyl-1H-pyrazol-4-yl)sulfonyl]-2-oxa-7-azaspiro[4.5]decane
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-[4-(3-fluorophenyl)benzoyl]-1,4-diazepan-5-one
N-[3-({[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]carbamoyl}amino)phenyl]-2-methoxyacetamide
3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-{[4-(methylsulfanyl)phenyl]methyl}piperidine
methyl[1-(1,2-oxazol-3-yl)ethyl]{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
2-[2-({methyl[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)phenyl]-6-(oxolan-2-yl)-3,4-dihydropyrimidin-4-one
N-[2-(5-methoxy-1H-indol-3-yl)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-methyl-6-{4-phenyl-1-[2-(pyridin-2-yl)ethyl]-1H-imidazol-5-yl}pyridine