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3-methyl-6-{3-[1-(2-phenylethyl)-1H-pyrazol-3-yl]phenyl}pyridazine
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,1-dimethylazepane-2-carboxamide
1-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-N-(thiolan-3-yl)piperidin-4-amine
N-[(2S,4R,6S)-2-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-6-(2-phenylethyl)oxan-4-yl]acetamide
(3aS,6aR)-3-[2-(4-fluorophenyl)ethyl]-5-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-methyl-4-[3-(5-methylfuran-2-yl)benzoyl]-1,4,9-triazaspiro[5.5]undecane
4-(1H-indol-3-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]butan-1-one
N-methyl-3-(5-methyl-1H-1,2,4-triazol-3-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}propanamide
1-(2-{[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl](methyl)amino}ethyl)piperidin-2-one
ethyl 3-{[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]amino}propanoate
N-[3-(1H-imidazol-1-yl)propyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
5-{1-[(2,4-difluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(1,4-dioxan-2-ylmethyl)-1-benzofuran-2-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-[2-(dimethyl-1,3-thiazol-4-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
3-(4-hydroxyphenyl)-4-(4-methoxy-2-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-ethoxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]propanamide
N-{3-oxo-3-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]propyl}methanesulfonamide
1-[2-(3-chlorophenyl)ethyl]-3-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]-2-(methoxymethyl)-6-methyl-1,4-dihydropyridin-4-one
N-{1-[(cyclopropylcarbamoyl)methyl]piperidin-4-yl}-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-phenoxy-1-(4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazin-1-yl)propan-1-one
methyl (2S,3S)-2-{[1-cyclohexyl-5-(methylcarbamoyl)-4-oxo-1,4-dihydropyridin-3-yl]formamido}-3-methylpentanoate
1-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]-2-[methyl(pyridin-2-ylmethyl)amino]ethan-1-one
(3R,9aR)-8-(3-methoxybenzoyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(3S,4S)-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-propylpyrrolidine-3-carboxylic acid
(2S,4S)-4-[5-(1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]-1-methylpyrrolidine-2-carboxylic acid
N-(2-hydroxyethyl)-6-methyl-N-[(2-methylphenyl)methyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
(3S,4R)-4-(2-methoxyphenyl)-1-(quinoline-3-carbonyl)pyrrolidine-3-carboxylic acid
1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-1,4-diazepan-6-ol
1-benzyl-8-(1H-imidazol-2-ylmethyl)-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-benzyl-3-methyl-8-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4,4-difluoro-N-{3-[(2-methylprop-2-en-1-yl)oxy]phenyl}piperidine-1-carboxamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N,1-dimethyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{[(8-chloro-4-hydroxyquinolin-2-yl)methyl](methyl)amino}-1λ6-thiane-1,1-dione
3-cyclopropyl-6-[(4-fluoro-2-methylphenyl)methyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
(2S,4R)-4-[(cyclohexylmethyl)amino]-1-(2,3-dihydro-1H-inden-2-yl)-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
1-ethyl-4-(3-methyl-3-phenylpiperidine-1-carbonyl)-1,2-dihydropyridin-2-one
4-(4-methanesulfonylphenyl)-3-methylpyridine
5-[({2-methylthieno[2,3-d]pyrimidin-4-yl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
N,2-dimethyl-N-(2-methylprop-2-en-1-yl)-6-(piperidin-3-yl)pyrimidin-4-amine
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-[2-oxo-3-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetamide
2-{5-[(3-methylthiophen-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1-propyl-1H-imidazole
1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
2-{2-[4-(6-methoxypyridin-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}-4-methyl-5,6,7,8-tetrahydroquinazoline
(2S)-2-[(2,6-dimethylquinolin-3-yl)formamido]-3-(4-hydroxyphenyl)propanoic acid
N,N,1-triethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(5-amino-1H-1,2,4-triazol-3-yl)-N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methylpropanamide
2-[4-(1-cyano-1-methylethyl)phenyl]-2-{methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}acetic acid
4-(4-{[(5,6-dimethylpyridin-3-yl)methyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)benzamide
(3S,4S)-1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
N-{[1-ethyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]methyl}-N-methylcyclopentanamine
2-(1-benzyl-3-oxopiperazin-2-yl)-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}acetamide