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3-{5-[(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)methyl]-4-phenyl-1H-imidazol-1-yl}propanoic acid
(2R,6S)-4-[1-(5-chloropyridine-3-carbonyl)piperidin-4-yl]-2,6-dimethylmorpholine
1-{1-[(6-methoxypyridin-3-yl)methyl]piperidin-4-yl}-2-phenylethan-1-ol
N-(2-methoxyethyl)-2-methyl-N-(3-phenylprop-2-yn-1-yl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-cyclopentyl-N-ethyl-4-(3-hydroxy-3-methylbutyl)benzamide
2-[2-methyl-4-(pyridin-4-yl)phenoxy]acetamide
ethyl 5-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1-(2,3-dimethylphenyl)-1H-pyrazole-4-carboxylate
N4-cyclopentyl-7-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-(1,3-benzothiazol-2-ylmethyl)-1-cyclohexyl-4-oxo-5-(pyrrolidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
4-(1-{1-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}ethyl)morpholine
4-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}-1-[(4-methylphenyl)methyl]piperazin-2-one
1-{[5-(methoxymethyl)furan-2-yl]methyl}-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
3-(6-chloropyridin-3-yl)-1-cyclohexyl-1-(2-hydroxyethyl)urea
N-[(3S,4R)-1-{2-[2-oxo-5-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetyl}-4-propylpyrrolidin-3-yl]acetamide
5-oxo-1-(pyridin-3-ylmethyl)-N-[2-(1,3-thiazol-2-yl)ethyl]pyrrolidine-3-carboxamide
N-[(3,4-difluorophenyl)methyl]-3-[1-(6-methylpyridine-2-carbonyl)piperidin-3-yl]propanamide
1'-(dimethyl-1,3-thiazole-5-carbonyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(2E)-N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-3-(3,4-dimethoxyphenyl)prop-2-enamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
N-(1-methylpiperidin-4-yl)-2-[3-(methylsulfanyl)phenyl]-N-(pyridin-4-ylmethyl)acetamide
N-(pyridin-3-ylmethyl)-4-[(2S)-2,4,5,5-tetramethylpiperazin-1-yl]pyridine-2-carboxamide
2-{4-[(4-methoxy-3-methylphenyl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
5-[4-(2-methoxyethoxy)phenyl]-6-methylpyridin-2-amine
3-methyl-6-{5-[1-(piperidin-4-yl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridazine
1-(2-methoxyphenyl)-N-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazole-4-carboxamide
6-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
4-(benzyloxy)-1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
5-(2,3-dihydro-1-benzofuran-7-yl)-3-(2-phenylethyl)-1H-1,2,4-triazole
1-methyl-9-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)ethyl]-1,4,9-triazaspiro[5.5]undecan-5-one
2-hydroxy-1-[4-(5-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-4-(methylsulfanyl)butan-1-one
2-(3-ethoxyphenyl)-2-{methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}acetic acid
3-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-N-(2-methoxyethyl)propanamide
1-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-2-(3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
N3-{[4-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperidine-1,3-dicarboxamide
3-(2-fluorophenyl)-1-{[5-(prop-2-en-1-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}pyrrolidine
1-[1-(diphenylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-phenylazepane
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-(4H-1,2,4-triazol-4-yl)propanamide
[1-(cyclohex-1-ene-1-carbonyl)-4-[(3-methoxyphenyl)methyl]piperidin-4-yl]methanol
5-[2-(1H-imidazol-2-yl)phenyl]-3-(1-methyl-1H-imidazol-4-yl)-1,2,4-oxadiazole
2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-N-[1-(2-fluorophenyl)piperidin-4-yl]acetamide
11-{methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}-4-[(4-methylphenyl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-{[4-(3-cyclohexylpyrrolidine-1-carbonyl)-1,3-oxazol-2-yl]methyl}-1H-1,3-benzodiazole
(2S,4S)-4-amino-N-{[5-(2-chlorophenyl)furan-2-yl]methyl}-1-methylpyrrolidine-2-carboxamide
N-[(3S,4R)-1-[6-(hydroxymethyl)pyridine-2-carbonyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
3-(2-fluorophenyl)-1-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
N-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(2-fluorophenyl)methyl]-N-methylpiperidin-3-amine
1-(4-methoxyphenyl)-2-({3-propyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1H-imidazole
4-fluoro-2-hydroxy-N-methyl-N-[(3-methylpyridin-4-yl)methyl]benzamide
1-{5-[1-butyl-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-5-yl]-1H-pyrazol-3-yl}ethan-1-one
1-{3-[2-(3-methoxyphenyl)azetidine-1-carbonyl]phenyl}-5-methyl-1H-1,2,3,4-tetrazole