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1-(3,5-dimethylphenyl)-4-(5-methyl-2,3-dihydro-1H-indole-2-carbonyl)piperazin-2-one
2-[4-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-1-yl]-N-(1-methyl-1H-1,2,3-triazol-4-yl)acetamide
(3S,4R)-1-(2-aminopyrimidin-4-yl)-3-benzyl-4-methylpiperidin-4-ol
5-{3-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-3-oxopropyl}imidazolidine-2,4-dione
3-methyl-1-{1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-3-yl}butan-1-one
3-[2-(2-fluorophenyl)ethyl]-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
methyl 4-[4-(1-methyl-1H-pyrrole-2-carbonyl)piperazin-1-yl]benzoate
1-(2,3-dihydro-1H-inden-2-yl)-4-(1,3-thiazol-4-ylmethyl)piperazine
1-[(5-fluoro-2-methoxyphenyl)methyl]-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
4-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
1-methyl-6-(pyridin-4-yl)-N-(1,2,3,4-tetrahydronaphthalen-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl 2-({2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}amino)acetate
1-[(2,3-difluorophenyl)methyl]-4-[1-(oxane-4-carbonyl)pyrrolidin-3-yl]piperidine
4-[(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-2-yl)methyl]morpholine
6-methyl-2-(4-{[3-(methylsulfanyl)propyl]amino}piperidin-1-yl)pyridine-3-carbonitrile
2-(furan-2-yl)-2-oxo-N-[(2R)-oxolan-2-ylmethyl]acetamide
4-(4-fluorophenyl)-1-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]butan-1-one
N-{[1-(2-fluorophenyl)cyclopentyl]methyl}-1H-pyrazole-4-carboxamide
8-[3-(dimethylamino)benzoyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]cyclopentanamine
5-methanesulfonyl-N-(2-methoxyethyl)-4-(piperidin-3-yl)pyrimidin-2-amine
N-({5-[(4-acetylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
4-({4-methyl-5-[1-(piperidin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
4-[(6-ethoxypyridin-3-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-{[2-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]methyl}pyridine
2-[5-(5,6,7,8-tetrahydro-1,6-naphthyridine-6-carbonyl)-1H-pyrazol-3-yl]phenol
1-{2-[2-(3-fluoro-2,4-dimethylphenyl)-1H-imidazol-1-yl]ethyl}pyrrolidin-2-one
3-ethyl-N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)-1H-pyrazole-4-carboxamide
4-{5-[1-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-1H-imidazol-2-yl]pyrimidin-2-yl}morpholine
N,N-dimethyl-2-[6-(1H-pyrazol-1-yl)pyrimidin-4-yl]benzamide
N-ethyl-2-[4-(5-hydroxypyrazine-2-carbonyl)piperazin-1-yl]acetamide
2-(2-aminoethyl)-N-(2-methoxyethyl)-N-(oxolan-2-ylmethyl)quinazolin-4-amine
3-[(3-methylquinoxalin-2-yl)methyl]-1,3-diazinane-2,4-dione
8-[3-(4-methoxyphenyl)propanoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]propanamide
5-chloro-4,6-dimethyl-N-[3-(4-methylpiperazin-1-yl)propyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
1-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]-1-[(1R,2S,3S,4R,5S)-tricyclo[3.2.1.02,4]octane-3-carbonyl]piperidine
4-[4-({[1-(morpholin-4-yl)cyclohexyl]methyl}amino)piperidin-1-yl]-N-(pyridin-3-ylmethyl)benzamide
N-benzyl-2-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]acetamide
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-ethoxyethan-1-one
(1R,5R)-6-{[2-(methylsulfanyl)phenyl]methyl}-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
2-cyclohexyl-N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-1,3-benzoxazole-6-carboxamide
3-(azepan-1-ylmethyl)-1-[(3,4-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
7-[(3,4-difluorophenyl)methyl]-2-(furan-3-carbonyl)-2,7-diazaspiro[4.5]decane
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
2-[({5-[2-(4-fluorophenyl)azetidine-1-carbonyl]furan-2-yl}methyl)sulfanyl]pyrimidine
8-[(2R)-2-amino-2-phenylacetyl]-3-{3-[methyl(2-methylpropyl)amino]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one