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(3aR,7aS)-2-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
5-(propan-2-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-({5-[(2E)-but-2-en-2-yl]-4-phenyl-1H-imidazol-1-yl}methyl)-5-methylpyrazine
(1S,6R)-3-{2-[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]-1,3-thiazole-4-carbonyl}-3,9-diazabicyclo[4.2.1]nonane
3-(pentan-2-yl)-8-(pyrazine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[5-(2-ethylpyrimidin-5-yl)-4-phenyl-1H-imidazol-1-yl]acetic acid
6-[(diethylamino)methyl]-N-(2,3-dimethylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-({1-[2-methyl-2-(morpholin-4-yl)propyl]pyrrolidin-3-yl}methyl)methanesulfonamide
4-{4-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]piperidin-1-yl}-6-methylpyrimidin-2-amine
2-ethyl-5-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidine
2-(1-{1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-amine
7-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
dimethyl(2-{2-[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
N-(2-methoxyethyl)-4-{[2-(2-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-(1'-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)ethan-1-one
1-[3-(2-oxopyrrolidin-1-yl)propyl]-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-ethylbutan-1-one
4-(3,3-diphenylpiperidine-1-carbonyl)morpholine
2-[1-(cyclohexylmethyl)-4-[5-(methoxymethyl)furan-2-carbonyl]piperazin-2-yl]ethan-1-ol
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-[(1-phenyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(2-ethoxypyridin-3-yl)methyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
3,5-dimethoxy-2-{[methyl(thian-4-yl)amino]methyl}benzoic acid
(2S,4S)-N-ethyl-4-(2-phenylacetamido)-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}[(3-methylpyridin-4-yl)methyl]amine
3-(3-fluorophenyl)-5-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)-1,2,4-oxadiazole
1-tert-butyl-4-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
8-{[5-(thiophen-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1R,3S)-3-methoxy-7-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]-7-azaspiro[3.5]nonan-1-ol
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidin-2-amine
N,N-dimethyl-3-[3-(propan-2-yloxy)benzoyl]piperidine-1-sulfonamide
N-(3-methoxyphenyl)-3-[4-(trifluoromethyl)benzoyl]piperidine-1-carboxamide
(1S,5R)-6-(4-fluoro-3-methylbenzoyl)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
11-(4-methoxy-2,5-dimethylphenyl)-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
(3S,9aR)-3-[(2S)-butan-2-yl]-8-[(3,4-dimethylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(methylsulfanyl)-1-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
4-{2-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]morpholin-4-yl}-5,6,7,8-tetrahydroquinazolin-2-amine
methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl](3-phenylbutyl)amine
3-[(dimethylamino)methyl]-N-[3-fluoro-4-(trifluoromethyl)phenyl]-3-hydroxypiperidine-1-carboxamide
methyl 6-benzyl-2-(diethylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-(1-ethylpiperidin-3-yl)-7-fluoro-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
5-butyl-1'-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
7-[4-methoxy-3-(morpholin-4-yl)benzoyl]-2-oxa-7-azaspiro[4.5]decane
2,6-dihydroxy-N-(3-phenoxypropyl)benzamide
3-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-5,5-dimethyl-1,3-oxazolidine-2,4-dione
N-(2-ethoxyethyl)-3-{[(3-hydroxypyrrolidin-3-yl)methyl]sulfamoyl}benzamide
3-[4-(cyclopropylamino)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
2-{[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzonitrile
(3R,5S)-5-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}pyrrolidin-3-ol