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2-(4-{2-[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]ethyl}piperazin-1-yl)pyrimidine
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-pentylpiperidine
3-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-1-[4-(oxolan-2-ylmethoxy)phenyl]urea
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-(4-methyl-2-oxo-1,2-dihydroquinolin-1-yl)-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]acetamide
6-(3-fluorophenyl)-N-methyl-N-[1-(pyridin-2-yl)propyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
8-(1-benzothiophen-2-ylmethyl)-1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-{pyrazolo[1,5-a]pyridine-3-carbonyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-[(2-{[3-(dimethylamino)pyrrolidin-1-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)methyl]-3,5-dimethyl-1,4-dihydropyridin-4-one
N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[2-(cyclohex-1-en-1-yl)ethyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
2,4-dimethoxy-N-({4-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzamide
3-(ethylsulfanyl)-1-(2-{[methyl(pyrazin-2-ylmethyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)propan-1-one
2-(dimethylamino)-2-(2-fluorophenyl)-N-(isoquinolin-5-ylmethyl)-N-methylacetamide
1-{1-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]piperidin-4-yl}-2-phenylethan-1-ol
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-(propan-2-yloxy)ethan-1-one
(3R,4R)-3-cyclobutyl-1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-methylpyrrolidin-3-ol
8-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-{5-[(4-methylpiperidin-1-yl)methyl]furan-2-carbonyl}-2-(trifluoromethyl)morpholine
(1S,5R)-6-(1H-indole-2-carbonyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-(3-fluoro-4-methylphenyl)-2-methyl-6-(4H-1,2,4-triazol-4-yl)pyridine
2-[5-(3,4-dihydro-2H-1-benzopyran-3-yl)-1,2,4-oxadiazol-3-yl]pyridine
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
3-(pyridin-4-yl)-7-thia-2,4,5-triazatricyclo[6.4.0.02,6]dodeca-1(12),3,5,8,10-pentaene
4-(2-methyl-1H-imidazol-1-yl)-1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}butan-1-one
ethyl 4-[3-(naphthalene-1-carbonyl)piperidin-1-yl]piperidine-1-carboxylate
3-[(3-methyl-1,2,4-oxadiazol-5-yl)(pyrrolidin-1-yl)methyl]pyridine
4-[1-({3-methyl-1-[2-(piperidin-1-yl)ethyl]-1H-pyrazol-4-yl}methyl)azetidin-3-yl]morpholine
6-ethyl-2-methyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]quinoline-4-carboxamide
N-(3-ethoxyphenyl)-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carboxamide
N-[(4-fluorophenyl)methyl]-1-methyl-5-{[2-methyl-2-(morpholin-4-yl)propyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-({[1-(4-butylphenyl)-1H-pyrazol-4-yl]methyl}amino)-2,3-dihydro-1λ6-thiophene-1,1-dione
N'-({1-[(2,3-dimethyl-1H-indol-7-yl)methyl]pyrrolidin-3-yl}methyl)ethanediamide
1-ethyl-4-[4-(2-methoxybenzoyl)piperazine-1-carbonyl]pyrrolidin-2-one
2-{1-[(3-methoxyphenyl)methyl]-4-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-{[(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)oxy]methyl}pyridine
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-3-(pyridin-3-yl)propan-1-one
1-cyclopentyl-4-(2,6-dimethylquinoline-4-carbonyl)piperazin-2-one
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methoxyethyl)acetamide
(1S,5R)-6-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(3-propyl-1H-pyrazole-4-carbonyl)piperidine
(1S,5R)-6-(cyclopropylmethyl)-3-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-5-yl}-3-[2-(propan-2-yloxy)ethyl]urea
4-{1-[1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]ethyl}morpholine
(2S)-N-[4-(3-methoxyphenyl)phenyl]-1-(1-methyl-1H-pyrrole-2-carbonyl)pyrrolidine-2-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-[2-(thiophen-2-yl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
1-(pyrimidin-2-yl)-4-[6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-1,4-diazepane
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(2-methylpropyl)-5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazole