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8-(4-methylpyrimidine-5-carbonyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(2-ethoxypyridine-3-carbonyl)-3-ethylpiperidine-3-carboxylic acid
3-(1,3-benzothiazol-2-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]propanamide
(2-{[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl](thiophen-3-ylmethyl)amino}ethyl)dimethylamine
2-(2-methoxyethyl)-9-(3-methyl-2-phenylbutanoyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]-2-(pyrrolidin-1-yl)benzamide
1-(2-methoxyethyl)-2-{[3-(3-methoxyphenoxy)azetidin-1-yl]methyl}-1H-imidazole
2-[5-cyclopropyl-4-(4-methylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-4-[2-(trifluoromethyl)phenyl]pyrimidine
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-3-phenoxypropanamide
dimethyl(2-{[(2-methylphenyl)methyl](1,3-thiazol-2-ylmethyl)amino}ethyl)amine
6-methyl-4-(trifluoromethyl)-1-[(3,4,5-trifluorophenyl)methyl]-1,2-dihydropyridin-2-one
1-{[4-(methylsulfamoyl)phenyl]methyl}-3-propylpiperidine-3-carboxylic acid
4,6-dimethyl-2-[3-(1H-pyrazol-3-yl)phenyl]pyrimidine
4-[({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]-N,N-dimethyl-1,3-thiazol-2-amine
(2S,4S)-4-amino-N,N-diethyl-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]pyrrolidine-2-carboxamide
3-({methyl[1-(3-phenylpropyl)piperidin-3-yl]amino}methyl)pyridin-2-amine
3-({methyl[(3-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)benzoic acid
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
6-ethyl-2-methyl-N-[3-(4-methylpiperazin-1-yl)butyl]quinoline-4-carboxamide
6-(dimethylamino)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methylpyridine-3-carboxamide
5-(2-butoxy-4-fluorophenyl)-3-cyclopropyl-1H-1,2,4-triazole
N-methyl-5-[(methylsulfanyl)methyl]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}furan-2-carboxamide
ethyl 2-[(3-{[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]carbamoyl}phenyl)amino]acetate
3-ethyl-1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-3-ol
N-benzyl-1-methyl-5-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(4aS,7aR)-1-cyclopentanecarbonyl-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[1-(4-methylpyridin-2-yl)propyl]-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
methyl 2-{[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]methyl}-1,3-oxazole-4-carboxylate
(2S)-2-({2-[(2,6-dichlorophenyl)methyl]-4-hydroxypyrimidin-5-yl}formamido)-3-methylbutanamide
4-{[(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)amino]methyl}-2,6-dimethylphenyl acetate
4-propyl-N-{2-[(trifluoromethyl)sulfanyl]ethyl}pyrimidine-5-carboxamide
N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]-4-(1H-1,2,3,4-tetrazol-1-yl)butanamide
6-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]piperazin-2-one
3-(2-{[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]amino}ethyl)-1,3-oxazinan-2-one
N-[1-(4-hydroxyphenyl)-2-methylpropan-2-yl]-2-(piperidin-4-yl)acetamide
(3R,7S,8aS)-7-{[(3-fluoro-4-methylphenyl)methyl]amino}-3-(2-methylpropyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
6-({[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amino)pyridine-3-carbonitrile
1-methyl-9-({2-phenylimidazo[1,2-a]pyridin-3-yl}methyl)-1,4,9-triazaspiro[5.5]undecan-5-one
(4aR,7aS)-1-acetyl-4-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl[(1-methyl-1H-imidazol-2-yl)methyl](2-phenylpropyl)amine
4-(5-hydroxypyrazine-2-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3R,4R)-N-[(4-chlorophenyl)methyl]-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidine-1-carboxamide
N,3,5,7-tetramethyl-N-(quinolin-5-ylmethyl)-1H-indole-2-carboxamide
2-cyclopropanecarbonyl-8-(pyrimidin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-cyclopropyl-7-fluoro-2-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]quinoline-4-carboxamide
1-(morpholin-4-yl)-3-{1-[2-(pyridin-2-ylsulfanyl)acetyl]piperidin-3-yl}propan-1-one
N-[4-(2,4-dimethyl-3-oxopiperazine-1-carbonyl)phenyl]-2-methylfuran-3-carboxamide
3-(3-chloro-1,2-oxazol-5-yl)-1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]propan-1-one
N,4-dimethyl-N-{[2-(2-methylpropoxy)phenyl]methyl}pyridine-3-carboxamide
(3aS,6aS)-2-(ethanesulfonyl)-5-[(2-fluoro-5-methoxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid