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5-(2-methoxyacetamido)-N-methyl-1-(2-phenylethyl)-N-(1H-pyrazol-5-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-(cyclopropylmethyl)-1-{1,3-dioxo-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}-N-propylpiperidine-3-carboxamide
{[(3S,4R)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}[(2-chlorophenyl)methyl]methylamine
N-(2-methoxyethyl)-2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[methyl(pyridin-3-ylmethyl)amino]methyl}piperidin-2-one
dimethyl({[(1R,5S,6S)-3-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-azabicyclo[3.1.0]hexan-6-yl]methyl})amine
2-[(3,5-dichloropyridin-4-yl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(2,6-dimethoxyphenyl)methyl]-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)piperidin-4-amine
6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-(pyrazine-2-carbonyl)-1,4-diazepan-2-one
7-methyl-3-[(3-methylquinoxalin-2-yl)methyl]-3,7,11-triazaspiro[5.6]dodecan-12-one
{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
4-(2,3-dimethoxyphenyl)-1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,3-triazole
4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-methyl-1-[(4-methylphenyl)methyl]piperazin-2-one
4-chloro-2-hydroxy-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-5-(furan-2-yl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-methoxy-N-{1-[1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(3-methylpyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3S,5R)-5-({5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyrrolidin-3-ol
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2-(phenylamino)pyrimidine-5-carboxamide
5-(1H-indol-1-ylmethyl)-N-[1-(pyridin-4-yl)propyl]-1H-pyrazole-3-carboxamide
2-[2-methyl-4-(pyrimidin-5-yl)phenoxy]acetamide
N6-cyclopentyl-N5-ethyl-N5-[2-(1H-pyrazol-1-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
3-methyl-7-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-benzyl-9-[2-(methylsulfanyl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
ethyl 2-{1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidin-2-yl}acetate
6-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
(3aR,5R,6S,7aS)-2-[1-(1-phenylethyl)-1H-1,2,3,4-tetrazol-5-yl]-octahydro-1H-isoindole-5,6-diol
5-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
1-{2-cyclooctyl-2,7-diazaspiro[4.5]decan-7-yl}-2-methoxyethan-1-one
5-amino-N-[(3R,5S)-5-(diethylcarbamoyl)-1-(furan-2-ylmethyl)pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
5-({3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)-2-(methoxymethyl)pyrimidine
N-butyl-N-ethyl-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-{[5-(1-cyclohexylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidin-4-ol
3-(1H-1,3-benzodiazol-2-yl)-N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)propanamide
(2E)-N-({7-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-(thiophen-2-yl)prop-2-enamide
(3aS,6aS)-2-cyclobutanecarbonyl-5-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-cyclohexyl-3-(cyclopropylmethyl)-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-(3-{[2-(2-methoxyethyl)piperidin-1-yl]methyl}-1H-indol-1-yl)propanamide
4-{[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}benzonitrile
5-(4-{[(benzylsulfamoyl)amino]methyl}piperidin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
1-(carbamoylmethyl)-N-[(4-fluorophenyl)(pyridin-4-yl)methyl]piperidine-4-carboxamide
2-({[1-(2-cyclohexylethyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}(methyl)amino)-N-methylacetamide
methyl 1-{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}piperidine-4-carboxylate
9-methoxy-10-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
N-{[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]methyl}-4-methylbenzene-1-sulfonamide
3-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-(2,3-dihydro-1H-inden-4-yl)urea