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N-[(3S,4R)-1-(1H-indole-2-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
4-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-7-fluoro-1,2-dihydroquinolin-2-one
2-methyl-2-[4-(morpholin-4-yl)-2-{[2-(oxan-2-yl)ethyl]amino}pyrimidin-5-yl]propanoic acid
4-({2-[1-(4-chlorobenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-(2-methoxy-4-methylphenoxymethyl)-N-methyl-N-(oxolan-2-ylmethyl)-1,3-oxazole-4-carboxamide
1-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-(propan-2-yloxy)propan-1-one
3-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chlorophenyl)urea
4-{3-[(4-methoxyphenyl)methyl]-5-(1-methylpiperidin-2-yl)-1H-1,2,4-triazol-1-yl}-2-methylpyridine
N-cyclopropyl-5-methyl-4-[(1,2,3,4-tetrahydronaphthalen-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
N-[3-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)carbamoyl}amino)-4-fluorophenyl]propanamide
4-{[3-(azepane-1-carbonyl)-1-ethyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}adamantan-1-ol
N,3,5-trimethyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-1H-indole-2-carboxamide
N-(3-chloro-4-fluorophenyl)-3-[1-(oxolane-3-carbonyl)piperidin-4-yl]propanamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-(2,3-dihydro-1H-inden-2-yl)-4-(piperidin-4-ylmethyl)-1,4-diazepane
methyl 4-[(2-{[methyl({[2-(trifluoromethyl)phenyl]methyl})amino]methyl}quinazolin-4-yl)amino]butanoate
4-(2,2-diphenylethyl)-3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]piperazin-2-one
1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(4-methoxybenzoyl)piperazine
1-[(4-chloro-3-fluorophenyl)methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
1-[4-(hydroxymethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]-2-(phenylsulfanyl)ethan-1-one
2-{[(4-hydroxy-5,8-dimethylquinolin-2-yl)methyl]amino}-N-methylethane-1-sulfonamide
4-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}piperazine-1-sulfonamide
6-(6-hydroxyhexyl)-3,4-dihydroquinazolin-4-one
4-chloro-6-[6-(methoxymethyl)pyrimidin-4-yl]-1-(prop-2-en-1-yl)-1H-1,3-benzodiazole
2-(4-methoxyphenoxymethyl)-N-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
[(3S,5R)-5-[(dimethylamino)methyl]-1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)piperidin-3-yl]methanol
N-{3-[({[1-(2-methoxyethyl)piperidin-3-yl]methyl}(methyl)carbamoyl)amino]phenyl}-N-methylacetamide
1-(2-methanesulfonylethyl)-4-(2-phenylpropyl)-1H-1,2,3-triazole
6-methyl-4-{4-[(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N-[2-(3-fluorophenyl)ethyl]-3-azaspiro[5.5]undecan-9-amine
N3-cyclohexyl-1-cyclopropyl-N5-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-(4-{[3-(dimethylamino)pyrrolidin-1-yl]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
5-[1-(3,6-dimethylpyrazin-2-yl)piperidin-4-yl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
3-methyl-1-(4-{5-[1-(1H-pyrazol-1-yl)propyl]-1,2,4-oxadiazol-3-yl}phenyl)-1H-pyrazol-5-amine
1-[(2-{[(5-cyclobutyl-1,3,4-oxadiazol-2-yl)amino]methyl}phenyl)methyl]pyrrolidin-2-one
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
2-[4-(1,3-benzoxazol-2-yl)-1-[(4-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-[3-(2-oxopyrrolidin-1-yl)propanoyl]-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-(9-methyl-9H-carbazol-3-yl)ethan-1-one
3-(morpholine-4-carbonyl)-1-propyl-5-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-4,5,6,7-tetrahydro-1H-indazole
N-(2,3-dihydro-1H-inden-5-yl)-4-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
8-cyclopropanecarbonyl-2-[(4-fluoro-2-methylphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-methyl-4-(2-{[6-(piperidin-1-yl)pyrimidin-4-yl]oxy}hex-5-en-1-yl)-1,4-diazepane
1-(azepan-1-yl)-3-{3-[(cyclopentylamino)methyl]phenoxy}propan-2-ol
N-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(pyridin-4-yl)acetamide
1-[2-(3-fluorophenyl)ethyl]-N-methyl-N-(naphthalen-1-ylmethyl)-6-oxopiperidine-3-carboxamide
2-[(1-ethyl-1H-imidazol-2-yl)methyl]-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
5-{[benzyl(methyl)amino]methyl}-N-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1,2-oxazole-3-carboxamide
5-chloro-6-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}pyridine-3-carboxylic acid
N-(2-hydroxyethyl)-1-[1-(3-phenylpropyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide