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N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(1H-pyrazol-1-yl)butanamide
N3-(1-benzylpyrrolidin-3-yl)-N5-ethyl-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-[(3,4-dimethoxyphenyl)methyl]-3-(1-methoxypropan-2-yl)-1-phenylurea
4-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]morpholine-2-carboxamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
2-(dimethylamino)-1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-2-(3-methylphenyl)ethan-1-one
1,3-dimethyl-N-{[1-(4-methylpiperazin-1-yl)cyclohexyl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
4-[4-(pyrrolidine-1-carbonyl)phenoxy]-1-[2-(4H-1,2,4-triazol-4-yl)ethyl]piperidine
2-(5-fluoro-2-methylphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
2-{4-[2-(2-aminoethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl]piperazin-1-yl}pyridine-3-carbonitrile
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-4-hydroxy-2-(phenoxymethyl)pyrimidine-5-carboxamide
5-hydroxy-1,2-dimethyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1H-indole-3-carboxamide
1-[4-chloro-2-(trifluoromethyl)phenyl]-3-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
N-methyl-3-[N-methyl-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamido]butanamide
4-methyl-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}pentan-1-one
4-[2-(2-methoxyphenoxy)-2-methylpropanoyl]-1-methylpiperazine-2-carboxylic acid
2-amino-6-(2-amino-4-methyl-1,3-thiazol-5-yl)-4-[2-(propylamino)pyrimidin-5-yl]pyridine-3-carbonitrile
5-(1H-imidazol-2-yl)-2-phenoxypyridine
1-[4-({[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}methyl)thiophen-2-yl]ethan-1-one
2-(3-{2-methyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl}piperidin-1-yl)acetamide
5-[2-(methylsulfanyl)ethyl]-1-(oxan-4-ylmethyl)-4-phenyl-1H-imidazole
5-acetyl-N-[(3-methyl-1H-pyrazol-5-yl)methyl]thiophene-2-carboxamide
1-(1,2-oxazolidin-2-yl)-2-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N'-(adamantan-1-yl)-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]propanediamide
2,7-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]imidazo[1,2-a]pyridine-3-carboxamide
4-({5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,2-dihydroisoquinolin-1-one
N-methyl-3-[methyl(1-methylpyrrolidin-3-yl)amino]-N-(quinolin-5-ylmethyl)propanamide
1'-[1-(2-methylpropyl)-5-oxopyrrolidine-3-carbonyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-(2,4-dimethoxyphenyl)-2-[2-(pyrrolidin-1-ylmethyl)-4-(thiophen-2-yl)phenoxy]acetamide
1-[1'-(4-fluoro-2-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
N-[(3R,4R)-3-hydroxy-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-4-yl]pyridine-3-carboxamide
N-[2-(pyridin-4-yl)ethyl]-3-{[(3R)-pyrrolidin-3-yl]sulfamoyl}benzamide
N-{3-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-3-oxopropyl}methanesulfonamide
5-(4-chlorophenoxy)-4-(1H-imidazol-2-yl)-1,3-dimethyl-1H-pyrazole
N-(2-hydroxyethyl)-3-[5-(2-methoxyethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
8-[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazole
N-(3-hydroxybutyl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
4-ethyl-1-methyl-3-({1-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl (3aR,6aR)-2-[(2-hydroxyphenyl)methyl]-5-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylate
2-(methylamino)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1,3-thiazole-4-carboxamide
methyl (2S,4S)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(3,4-difluorophenyl)methyl]pyrrolidine-2-carboxylate
5-methyl-N-[(2-phenoxypyridin-3-yl)methyl]thiophene-2-sulfonamide
4,4-difluoro-N-(1-propyl-1H-1,3-benzodiazol-5-yl)piperidine-1-carboxamide
5-[2-(3,4-dimethylphenoxy)ethyl]pyridine-3-carboxamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-N-(4-methoxyphenyl)piperidin-3-amine
3-methyl-8-{2-[methyl(phenyl)amino]acetyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)(4,5,6,7-tetrahydro-2H-indazol-3-ylmethyl)amine