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(1R,2S)-1-({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-2,3-dihydro-1H-inden-2-ol
8-(cyclopropanesulfonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
(2R,6S)-4-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-2,6-dimethylmorpholine
7-[(4-fluorophenyl)methyl]-2-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-(2-ethoxyethyl)-2-(6-methoxynaphthalen-2-yl)morpholine
1-{4-[3-(piperidine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]piperazin-1-yl}ethan-1-one
N-[4-(dimethylamino)phenyl]-2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
4-(3-methylfuran-2-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2,3-dimethyl-5-phenyl-N-(3,3,3-trifluoropropyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-butyl-N-[(3-methoxyphenyl)methyl]-2-methyl-1H-imidazole-4-carboxamide
N-ethyl-2-(morpholin-4-yl)-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}acetamide
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(2-propyl-1H-1,3-benzodiazol-1-yl)propanamide
2-[3-(2-methoxyphenoxy)azetidin-1-yl]-4-methyl-1,3-thiazole
4-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-methyl-1-(2-methylpropyl)piperazin-2-one
8-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
(2S,4S,5R)-5-(2-chlorophenyl)-1,2-dimethyl-4-(pyrrolidine-1-carbonyl)pyrrolidine-2-carboxylic acid
N-[(2,4-dimethoxyphenyl)methyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
8-(5-amino-1H-pyrazole-3-carbonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
1-(4-methyl-3-phenylpiperazine-1-carbonyl)cyclopropan-1-amine
2-(2-cyclopropylpyrimidine-5-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-2-(dimethylamino)-2-(4-methylphenyl)acetamide
4-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]-2-(trifluoromethyl)morpholine
3-[(cyclopropylcarbamoyl)methyl]-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-(2-{[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}ethyl)piperidin-2-one
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-[(3-methylphenyl)methyl]piperidin-3-ol
4-(4-chlorophenyl)-N-[(3S)-2-oxo-1,2,3,4-tetrahydroquinolin-3-yl]butanamide
3-{1-[(5-chlorofuran-2-yl)methyl]piperidin-4-yl}-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
2-(2-fluorophenyl)-1-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
8-(4-aminopyridine-2-carbonyl)-2-cyclopentyl-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
2-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-fluoropyridine
2-[4-(1,3-benzothiazol-2-ylmethyl)-1-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
1-[4-({[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]amino}methyl)piperidin-1-yl]-2-methylpropan-1-one
1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-4-methylpentane-1,2-dione
4-(5-fluoro-2-methylbenzoyl)-3-methyl-1-(2-methylpropyl)piperazin-2-one
1-[5-(hydroxymethyl)furan-2-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
ethyl[(1-ethyl-1H-imidazol-2-yl)methyl]({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amine
5-{2-[4-(4-methoxyphenyl)-2-methyl-3-oxopiperazin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
N-cyclopropyl-2-({1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}oxy)-4-methoxybenzamide
4-(piperidin-1-yl)-1-[3-(pyridin-3-yl)azetidin-1-yl]butan-1-one
{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
1-cyclohexyl-N-[(3,5-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-{imidazo[1,2-a]pyridin-2-ylmethyl}-6-methyl-3,4-dihydroquinazolin-4-one
N-({5,7-dimethylimidazo[1,2-a]pyridin-2-yl}methyl)-3-(1-methylpiperidin-2-yl)propanamide
4-[(diethylamino)methyl]-5-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]furan-2-carboxamide
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]pyrrolidine-3-carboxamide