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N-{[7-(2-cyclopentyl-2-phenylacetyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzamide
1-(furan-2-ylmethyl)-4-[4-(3-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]piperidine
(3R,5S)-5-(3-fluorophenoxymethyl)-N-[2-(1H-imidazol-4-yl)ethyl]-1-(pyridin-4-ylmethyl)piperidine-3-carboxamide
N-[1-(hydroxymethyl)cyclopentyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-oxazole-3-carboxamide
N-[(2-chlorophenyl)methyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-(prop-2-en-1-yl)acetamide
4-hydroxy-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
N-[(3S,4R)-4-(propan-2-yl)-1-[4-(trifluoromethyl)benzenesulfonyl]pyrrolidin-3-yl]acetamide
3-chloro-4-({1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
2-(pyridin-4-yl)-N-[1-(pyrimidin-4-yl)ethyl]quinoline-4-carboxamide
1-{2-hydroxy-3-[2-({[(1-hydroxycyclohexyl)methyl]amino}methyl)-4-methoxyphenoxy]propyl}piperidin-4-ol
3-(4-hydroxyphenyl)-1-[4-(2-methoxyethyl)piperazin-1-yl]-2-phenylpropan-1-one
N-{3-hydroxy-1-[4-(propan-2-yl)phenyl]propyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
5-(oxan-3-yl)-2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-[3-(4-fluorophenoxymethyl)-5-(1,2-oxazol-3-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
(4aS,7aR)-1-(2,6-dimethoxypyridine-3-carbonyl)-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3R,4R)-4-ethyl-1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)piperidine-3,4-diol
3-[2-(4-fluorophenyl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indazole
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2,4-dimethylpyrimidine-5-carboxamide
N-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1H-1,2,3-triazole-5-carboxamide
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-5-ethyl-N-methylpyrazolo[1,5-a]pyrimidin-7-amine
N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-benzothiophene-2-carboxamide
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]-2-propylpyridine-4-carboxamide
2-ethoxy-5-(2-{[2-(pyrrolidin-1-yl)ethyl]amino}pyrimidin-4-yl)benzoic acid
8-[2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[4-(dimethylamino)oxan-4-yl]methyl}-1,7-dimethyl-1H-indole-2-carboxamide
(3aR,6aR)-2-(2-chloro-4-fluorobenzoyl)-5-(cyclobutylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2S,4S)-4-amino-1-[2-(3-chlorophenoxy)acetyl]pyrrolidine-2-carboxylic acid
(3S,4S)-4-({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)-1-(propan-2-yl)pyrrolidin-3-ol
3-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)pyridin-2-ol
N3-tert-butyl-N5-[(4-chlorophenyl)(phenyl)methyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-amino-6-methyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}pyrimidine-4-carboxamide
[5-(1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methanol
2-{1-cyclohexyl-5-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-1H-1,2,4-triazol-3-yl}acetamide
4-(4-{[(3-hydroxypropyl)amino]methyl}phenyl)benzonitrile
1-(4-{[2-(dimethyl-1,3-thiazol-2-yl)ethyl]amino}-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
4-{2-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]ethyl}-2-ethyl-1,3-thiazole
(2S,4R)-N,1-dimethyl-4-({5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}amino)pyrrolidine-2-carboxamide
4-ethyl-3-[1-(5-methyl-1H-indazole-3-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[(1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-yl)oxy]pyrimidine
2,3-dimethyl-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]quinoxaline-6-carboxamide
3-(piperidin-1-ylmethyl)-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-ol
3-(hydroxymethyl)-1-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methyl)piperidin-3-ol
8-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]acetamide
ethyl 4-benzyl-1-(3-phenylprop-2-yn-1-yl)piperidine-4-carboxylate
4-hydroxy-1-[(2-methylphenyl)methyl]piperidine-4-carboxylic acid
3-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,3-dichlorophenyl)urea
2-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1,2-dihydroisoquinolin-1-one
2,7,8-trimethyl-N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]quinoline-4-carboxamide
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]acetamide