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5-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[(2-methoxyphenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazole
3-(3-hydroxyquinoxalin-2-yl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]propanamide
5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-2-(4H-1,2,4-triazol-4-yl)pyridine
2-oxo-N-{[1-(pyridin-2-ylmethyl)piperidin-3-yl]methyl}butanamide
methyl (2S)-2-{[1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidin-4-yl]formamido}-2-phenylacetate
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-4-yl}propanamide
6-(2,4-dimethylbenzoyl)-2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
3-tert-butyl-5-{[5-(furan-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
1-(4-ethoxy-2-fluorophenyl)-3-[(2S)-pyrrolidin-2-ylmethyl]urea
N-(3-methoxypropyl)-6-[4-(thiophen-2-ylmethyl)piperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
4-(1-methyl-1H-imidazol-2-yl)-1-(1,3-thiazol-2-ylmethyl)piperidine
3-chloro-6-(4-{4-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-1,2,3-triazol-1-yl}piperidin-1-yl)pyridazine
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
4-[3-(azepane-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]-1,4-diazepane-1-carbaldehyde
6-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine-2,4-diamine
(1-{1-[(2,3,4-trimethoxyphenyl)methyl]piperidin-3-yl}piperidin-4-yl)methanol
4-cyclopropyl-6-(4-methanesulfonylphenyl)pyrimidine
2-(pyridin-2-yl)-5-[4-(pyridin-2-yl)piperazine-1-carbonyl]pyrimidin-4-ol
N-[2-(azepane-1-carbonyl)phenyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-phenyl-N-({1-[2-(phenylsulfanyl)acetyl]piperidin-3-yl}methyl)benzamide
1-[4-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-3-methyl-3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]urea
(3S,4R)-1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
3-{[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}benzoic acid
N-[2-(cyclohex-1-en-1-yl)ethyl]-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamide
2-[3,5-bis(trifluoromethyl)phenyl]-4-hydroxy-N-methyl-N-(2-methylpropyl)pyrimidine-5-carboxamide
1-{[4-(hydroxymethyl)oxan-4-yl]methyl}-3-[3-(1H-imidazol-5-yl)phenyl]-1-methylurea
(2R,3R,6R)-3-(4-fluorophenyl)-5-(pyridazine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-methyl-4-(3-{4-[(methylsulfanyl)methyl]piperidine-1-carbonyl}phenyl)butan-2-ol
3-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-(propan-2-yl)pyrrolidine
4-(ethoxymethyl)-1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidine
3-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
2-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-3-yl]-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
6-cyclopentyl-N-[2-(1H-imidazol-2-yl)ethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-({1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}methyl)-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(3-methoxypyrazin-2-yl)-5-[2-(piperidin-2-yl)ethyl]phenol
(3R)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
[(2S)-1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl]methanol
(1R,3S)-3-(2-aminoethoxy)-7-[2-(difluoromethoxy)benzoyl]-7-azaspiro[3.5]nonan-1-ol
methyl 5-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-5-oxopentanoate
4-{4-[(2-ethylmorpholin-4-yl)methyl]phenyl}-2-methylbutan-2-ol
methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}){[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}amine
1-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3,3-dimethylbutan-1-one
2-(2,5-dioxoimidazolidin-1-yl)-N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
N-{2-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]-2-oxoethyl}methanesulfonamide
4-fluoro-1-({5-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)piperidine
N-cyclohexyl-N-[2-(dimethylamino)ethyl]-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-(2-methylpropyl)-1-[(1s,4s)-4-acetamidocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-(oxolan-2-ylmethyl)-5-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}pyrimidin-2-amine
3-[3-(4-phenyl-5-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-imidazol-1-yl)propyl]pyridine