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N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
N-{2-[methyl(2-phenylethyl)amino]ethyl}-4-(pyridin-3-yl)pyrimidin-2-amine
(2-{1-[(5-fluoro-2-methoxyphenyl)methyl]piperidin-2-yl}ethyl)dimethylamine
2-[3-(2-methyl-1H-imidazol-1-yl)propyl]-5-(4-methylpiperazin-1-yl)-2,3-dihydropyridazin-3-one
2-(2,3-dimethoxyphenyl)-4-methoxypyrimidine
N-methyl-2-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethane-1-sulfonamide
3-{[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl](methyl)amino}-N-methylbutanamide
1-[2-(dimethylamino)-4-({[3-(pyrrolidin-1-yl)phenyl]methyl}amino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-methyl-5-{[2-(2,4,7-trimethyl-1H-indol-3-yl)acetamido]methyl}furan-2-carboxamide
N-(2-hydroxyethyl)-5-(1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}pyrrolidin-2-yl)thiophene-2-carboxamide
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-1H-pyrazole-4-carboxamide
1-{2-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
2-(ethylamino)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}pyrimidine-5-carboxamide
N-[(5-methylthiophen-2-yl)methyl]-3-(2-oxopiperidin-1-yl)-N-(pyridin-4-ylmethyl)propanamide
5-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-2,3-dihydro-1H-indol-2-one
2-(morpholin-4-yl)-1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,3-benzodiazole
5-ethyl-1'-(5,6,7,8-tetrahydroquinoline-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
ethyl 4-(cyclopropylmethyl)-1-{[4-(methylsulfanyl)phenyl]methyl}piperidine-4-carboxylate
8-benzyl-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-5-[(2-phenyl-1,3-oxazol-4-yl)methyl]-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2,2,2-trifluoroethyl)acetamide
2-{N-methyl-1-[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]formamido}-2-(thiophen-2-yl)acetic acid
5-[4-(piperidin-1-ylmethyl)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-3-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
5-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}-N-propylpyrimidin-2-amine
[(5-ethylfuran-2-yl)methyl]({[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl})amine
5-cyclopropyl-1-[4-(furan-2-yl)pyrimidin-2-yl]-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-1H-pyrazole-4-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetamide
2,6,8-trimethyl-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}quinoline-4-carboxamide
2-[1-methyl-4-(oxan-4-yl)-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl]acetic acid
9-methoxy-3-(5-phenylpentanoyl)-10-(thiomorpholine-4-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]-2-{4-oxo-3H,4H-thieno[3,2-d]pyrimidin-3-yl}acetamide
1-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-5-oxopyrrolidine-3-carboxylic acid
6-(1H-indol-5-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
4-{[(3S,5R)-1-(2-methylpropyl)-5-(pyrrolidine-1-carbonyl)piperidin-3-yl]methyl}morpholine
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-[2-(1H-pyrazol-4-yl)ethyl]-1,2,4-oxadiazole
4-[(2,5-difluorophenyl)methyl]-7-(2,3-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(isoquinolin-5-ylmethyl)-N-methyl-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
methyl N-{2-oxo-2-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}carbamate
8-(4-methoxycyclohexanecarbonyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
4-(4-methylphenoxy)-4-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]piperidine
N-methyl-3-(5-methylfuran-2-yl)-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
4-({1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}oxy)-N-(pyridin-4-ylmethyl)benzamide
1-[1-(cyclohexylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
(2S)-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-6-oxopiperidine-2-carboxamide
N-(2-fluorophenyl)-3-[1-(pyridin-4-ylmethyl)piperidin-3-yl]propanamide
2-[(1S,5R)-3-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
(3S,4S)-4-methyl-1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]piperidine-3,4-diol
N-(3-carbamoyl-4-methoxyphenyl)-4-(pyridin-3-ylmethoxy)piperidine-1-carboxamide
4-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-3-yl]-5-(2-fluorophenyl)-2-(pyridin-3-yl)pyrimidine