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1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(oxolane-2-carbonyl)piperazine
7-methyl-3-{5-[(4-methylpiperazin-1-yl)methyl]pyridin-2-yl}-1H-indole
1-(4-acetyl-1,4-diazepan-1-yl)-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}ethan-1-one
N-ethyl-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
N,N,2-trimethyl-4-{[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
dimethyl(1-{3-[3-(piperidine-1-carbonyl)pyridin-2-yl]phenyl}ethyl)amine
3-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]propanamide
2-[3-(furan-2-yl)-5-(morpholin-2-ylmethyl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
ethyl 4-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamido]piperidine-1-carboxylate
2-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-6-methylpyridine-3-carbonitrile
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-3-(3-methylphenyl)-1H-pyrazole-4-carboxamide
(2R,6S)-2,6-dimethyl-4-{1-[3-phenyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}morpholine
1-methyl-4-[5-(1H-1,2,3,4-tetrazol-1-ylmethyl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl]piperidine
1-(1,2,3,4-tetrahydroisoquinolin-2-yl)-3-(3-{[(thiophen-2-ylmethyl)amino]methyl}phenoxy)propan-2-ol
(1S,5R)-6-(cyclobutylmethyl)-3-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
5-(2,2-dimethyl-3-oxopiperazine-1-carbonyl)-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
[(3R,5R)-1-(5-methylpyridine-2-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[(5-methylpyrazin-2-yl)methyl]acetamide
1-(2-{[(5-chlorofuran-2-yl)methyl](methyl)amino}ethyl)piperidin-2-one
1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4-(3-methylpyridin-4-yl)-1,4-diazepane
N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]azetidin-3-yl}piperidine
N-(2,5-dimethylphenyl)-2-(2-methoxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
(4aR,8aR)-2-cyclopentanecarbonyl-7-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
4-(3-hydroxy-3-methylbutyl)-N-{[4-(hydroxymethyl)phenyl]methyl}benzamide
(1,4-dioxan-2-ylmethyl)(methyl){[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}amine
(5-{[7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]methyl}furan-2-yl)methanol
N-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-2-methyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
4-{[3-(2-hydroxyethyl)-4-[(4-methoxy-3-methylphenyl)methyl]piperazin-1-yl]methyl}-2-methoxyphenol
(furan-2-ylmethyl)(3-methylbut-2-en-1-yl)(thiophen-3-ylmethyl)amine
3-(1H-pyrazol-4-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}benzamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2,2-dimethylpropanamide
5-benzyl-4-(2-methoxyacetyl)-1-(2-phenylphenyl)piperazin-2-one
5-({3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)-2-(methylsulfanyl)pyrimidine
(4S)-1-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
N-methyl-3-(piperidine-1-carbonyl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrazine-2-carboxamide
1-(2-ethoxyethyl)-5-(4-ethyl-3-oxopiperazine-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-ethyl-N-(oxolan-2-ylmethyl)benzamide
3-methyl-N-{1-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
4-[(2,3-dihydro-1H-inden-2-yl)amino]-1-[2-(4-methoxyphenyl)ethyl]pyrrolidin-2-one
5-ethyl-2-methyl-N-[(5-methylpyrazin-2-yl)methyl]pyrimidin-4-amine
2-ethyl-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-methyl-1,3-oxazole-5-carboxamide
[(4-ethyl-1,3-thiazol-2-yl)methyl](4-methoxy-4-methylpentan-2-yl)amine
3-methoxy-2,2-dimethyl-N-[(2-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)propanamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}propanamide
5-[2-(2-hydroxyethyl)morpholine-4-carbonyl]-2-methyl-2,3-dihydro-1H-isoindole-1,3-dione
6-(2-aminoethyl)-N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-2-methylpyrimidin-4-amine
(3R,5S)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-N-[3-(morpholin-4-yl)propyl]-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide