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(1S,5R)-6-propyl-3-{2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(2-phenoxyethyl)piperazine
(4aS,8aR)-1-(carboxymethyl)-6-(5,6-dimethylpyrimidin-4-yl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
3-[4-(2-oxo-2,3-dihydro-1H-indol-1-yl)piperidin-1-yl]-N-(1,3-thiazol-2-yl)propanamide
(3R,5S)-N3-[2-(3-fluorophenyl)ethyl]-N5-(6-methylpyridin-3-yl)piperidine-3,5-dicarboxamide
6-oxo-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-1,6-dihydropyridine-2-carboxamide
4-{3-[4-(pyrrolidine-1-sulfonyl)phenyl]phenyl}-4H-1,2,4-triazole
N-(5-cyclobutyl-1,3,4-thiadiazol-2-yl)-4-(pyrimidin-2-yl)-1,4-diazepane-1-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(2-chlorophenyl)methyl]piperidin-3-ol
6-(2,3-dihydro-1-benzofuran-7-yl)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[(4-cyclopentylpyrimidin-2-yl)amino]-1-phenylethan-1-ol
7-{[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-methyl-2-{8-methyl-3-oxo-2,8-diazaspiro[4.5]decan-2-yl}-N-(1,3-thiazol-2-ylmethyl)acetamide
4-({4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidin-2-yl}amino)butan-1-ol
N-methyl-5-[(4-methylpiperazin-1-yl)methyl]-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
[1-(5-chloro-2-methoxybenzoyl)-3-(3-methoxypropyl)piperidin-3-yl]methanol
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(3R)-4-hydroxy-3-methylbutyl]-1H-pyrazole-3-carboxamide
2-(cyclopropylmethyl)-7-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-(hydroxymethyl)-1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]piperidin-4-ol
3-hydroxy-3-{[(1,2-oxazol-5-ylmethyl)amino]methyl}-1-(2-phenylethyl)piperidin-2-one
3-hydroxy-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-1-(2-phenylethyl)piperidin-2-one
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-methylpyridin-4-yl)methyl]acetamide
2-(3-chloro-4-hydroxyphenyl)-N-(3-hydroxypropyl)-N-[(5-methylthiophen-2-yl)methyl]acetamide
[(2S,6S)-4-(1H-imidazol-4-ylmethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
4-[(8-chloro-4-hydroxyquinolin-2-yl)methyl]-3-(2-hydroxyethyl)piperazin-2-one
4-[3-cyclopropyl-5-(1,4-dioxan-2-yl)-1H-1,2,4-triazol-1-yl]-2-methylpyridine
3-{[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl](prop-2-en-1-yl)amino}-1λ6-thiolane-1,1-dione
4-{[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl}-N-(trimethyl-1H-pyrazol-4-yl)benzamide
ethyl 3-(2-phenylethyl)-1-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxylate
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-[(4-methyl-1H-imidazol-5-yl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[(3R,4S)-4-cyclopropyl-1-[2-methyl-2-(morpholin-4-yl)propyl]pyrrolidin-3-yl]-2-methylpyrimidin-4-amine
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
8-[4-(4-methylpiperazin-1-yl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-[(3R,4R)-3-{[ethyl(2-hydroxyethyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-4-methylbenzene-1-sulfonamide
2-(2H-1,3-benzodioxol-5-yl)-N-[(2-propyl-1,3-thiazol-4-yl)methyl]acetamide
methyl 3-({[4-(4-fluorophenyl)phenyl]formamido}methyl)-5-(pyrazine-2-amido)benzoate
3-{1-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]piperidin-3-yl}benzoic acid
5-(azepane-1-carbonyl)-1-(butan-2-yl)-N-[(5-fluoro-2-methylphenyl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2-tert-butyl-4-hydroxy-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[(1-methyl-1H-imidazol-2-yl)methyl]benzamide
N-[(3-chlorophenyl)methyl]-3-[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]propanamide
N-methyl-5-({4-phenyl-5-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-imidazol-1-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
N-{1-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propanoyl]piperidin-4-yl}methanesulfonamide
1-(2-{1-[(5-methoxy-1H-indazol-3-yl)methyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
2-[(dimethylcarbamoyl)amino]-N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]acetamide
6-(2,5-dimethylfuran-3-yl)-7-methyl-2-(2-methylpiperidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-{2-[(dimethylcarbamoyl)methyl]phenyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carboxamide
2,5-dimethyl-3-[4-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperazin-1-yl]pyrazine