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1-(2H-1,3-benzodioxol-5-yl)-2-[5-(oxolan-2-yl)thiophen-2-yl]-1H-imidazole
methyl 5-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
3-{[ethyl(2-methoxyethyl)amino]methyl}-6-methoxy-1,2-dihydroquinolin-2-one
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-{3-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1H-pyrazol-1-yl}acetamide
N-(1-methyl-1H-pyrazol-3-yl)-2-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
4-[4-(2-methoxyphenyl)-1H-imidazol-2-yl]-1-[(2-methoxyphenyl)methyl]pyrrolidin-2-one
1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]({[2-(ethylsulfanyl)pyrimidin-5-yl]methyl})methylamine
4-(pyridin-3-ylmethyl)-N-[4-(trifluoromethyl)phenyl]-1,4-diazepane-1-carboxamide
N-benzyl-N-[(3-methylpyridin-2-yl)methyl]-2-(2-oxopiperidin-1-yl)acetamide
N,1-dimethyl-N-[2-(pyridin-2-yl)ethyl]-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[2-(diethylamino)ethyl]-N-ethyl-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
2-[2-(2-butyl-2,5-dihydro-1H-pyrrol-1-yl)-2-oxoethyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
1-[2-chloro-5-(trifluoromethyl)benzoyl]-3-(1H-imidazol-2-yl)piperidine
2-[4-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
(1S,5R)-6-[6-(methoxymethyl)pyridine-2-carbonyl]-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
1-[(4-methoxyphenyl)methyl]-4-(6-methoxypyrimidin-4-yl)piperazin-2-one
(3R,7S,8aS)-7-{[(2,4-difluorophenyl)methyl]amino}-3-[(1S)-1-hydroxyethyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
5-fluoro-2-[3-(piperidin-1-yl)pyrrolidine-1-carbonyl]phenol
1-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-(5-methyl-1,2-oxazol-3-yl)-N-[2-methyl-5-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]pyrrolidine-1-carboxamide
2-amino-4-[3-(2-hydroxyethoxy)phenyl]-6-(1H-indol-3-yl)pyridine-3-carbonitrile
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(3E)-N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-phenylbut-3-enamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-[(1-methyl-1H-imidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(3S)-N,N-dimethyl-1-(5-methyl-2-phenylfuran-3-carbonyl)azepan-3-amine
({4-[1-(cyclopropanesulfonyl)piperidin-2-yl]phenyl}methyl)dimethylamine
3-(1,2-oxazolidin-2-yl)-1-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]propan-1-one
N-(2-methylpropyl)-1-[(1s,4s)-4-{[(2-hydroxy-3-methoxyphenyl)methyl]amino}cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
ethyl({[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
2-{1-cyclohexyl-4-[(1-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
2,7-dimethyl-N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-tert-butyl-2-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}butanamide
{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
5-[2-(cyclohexylmethyl)morpholine-4-carbonyl]quinoxaline
methyl 7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxylate
N-(4-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-4-oxobutan-2-yl)acetamide
6-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-4-(pyridin-2-yl)pyrimidine
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[3-(2-fluorophenyl)-1H-pyrazol-1-yl]acetamide
1-{2-methylpyrido[2,3-d]pyrimidin-4-yl}-4-(1,3-thiazol-2-yl)piperazine
N-(2-chloro-5-methylphenyl)-3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazine-1-carboxamide
2-(3-methoxypropyl)-8-[4-(1H-pyrazol-4-yl)butanoyl]-2,8-diazaspiro[4.5]decan-3-one
6-[(3S)-3-ethylmorpholine-4-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
3-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1-ethyl-6-methyl-1,2-dihydropyridin-2-one
5-(2-methyl-4-phenylpiperazine-1-carbonyl)-2-(thiophen-2-yl)pyrimidin-4-ol
N-(1-benzylpyrrolidin-3-yl)-3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]propanamide
4-(1H-imidazol-1-ylmethyl)-1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-ol