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2-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]propane-1,3-diol
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)pyridine-3-carboxamide
8-methoxy-2-(thiophen-2-yl)quinoline
N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
3-(1-methylpiperidin-4-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]propanamide
5-(3-methylbut-2-en-1-yl)-1'-(pyrrolidine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-fluoro-2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-N,N-dimethylpyrimidin-4-amine
5-[(dimethylsulfamoyl)amino]-N-(1H-indol-2-ylmethyl)-1-methyl-2-(2-methylpropyl)-1H-1,3-benzodiazole-7-carboxamide
methyl[1-(1,2-oxazol-3-yl)ethyl][(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amine
3,6,7-trimethyl-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1-benzofuran-2-carboxamide
2-[({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)amino]propan-1-ol
1-[3-({[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}methyl)piperidin-1-yl]ethan-1-one
[1-(5-ethyl-2-methylpyrimidin-4-yl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
2-ethyl-4-(1-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-4-phenyl-1H-imidazol-5-yl)pyrimidine
(5E)-5-({3-chloro-4-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methoxy]phenyl}methylidene)imidazolidine-2,4-dione
(3-{[1-(3-phenyl-1,2-oxazole-5-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
1-[3-methyl-1-(4-methylphenyl)-1H-1,2,4-triazol-5-yl]-1-phenylethan-1-ol
3-[(1-cycloheptylpiperidin-3-yl)sulfamoyl]benzoic acid
(1R,2S,6R,7S)-4-[3-(piperidine-1-carbonyl)pyridin-2-yl]-4-azatricyclo[5.2.2.02,6]undecane
6-methyl-2-[(2-methylphenyl)methyl]-4-oxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-cyclopropyl-9-[4-(hydroxymethyl)benzoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]-2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]acetamide
N-benzyl-4-hydroxy-4-(hydroxymethyl)-N-methylpiperidine-1-sulfonamide
2-cyclohexyl-5-{5-[(1-methyl-1H-imidazol-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyrimidine
5,7-dimethyl-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
8-methoxy-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-1-methyl-1,4,9-triazaspiro[5.5]undecane
2-(ethylamino)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]pyrimidine-5-carboxamide
7-(3-chlorophenyl)-4-[2-(1H-pyrazol-4-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(4aS,8aR)-6-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
5-cyclopropanecarbonyl-1'-(dimethyl-1,2-oxazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(dimethylamino)ethan-1-one
1-{2-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]phenyl}-1,3-diazinane-2,4-dione
2-{2-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethoxy}ethan-1-ol
(2S)-1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-3-methyl-2-(methylamino)butan-1-one
(2Z)-2-fluoro-1-{3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}-3-phenylprop-2-en-1-one
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[3-(phenylamino)piperidin-1-yl]propan-1-one
N-{2-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]ethyl}-3-methylpyridin-4-amine
(1S,5R)-3-benzyl-6-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
8-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(2R,3R,6R)-5-[(5-ethylpyridin-2-yl)methyl]-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-(2,3-difluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(4-{3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)ethan-1-amine
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
(1R,5S,6R,7S)-3-(2-aminoethyl)-4-oxo-N-(pyridin-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]decane-6-carboxamide
4-chloro-5-[({imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)amino)methyl]-N,N-dimethyl-1,3-thiazol-2-amine
4-[(2-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-3-yl}-1H-imidazol-1-yl)methyl]pyridine
N-[3-(3-methoxyphenyl)phenyl]-1-(thian-4-yl)piperidine-4-carboxamide
1-[1-(hydroxymethyl)-9-(2-phenylethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-2-methoxyethan-1-one
1-(2-methylpropyl)-4-oxo-N3-(2-phenylpropyl)-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide