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2-(2,3-dihydro-1H-inden-1-yl)-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}acetamide
N-(1-{2-[(2-methoxyethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-yl)methanesulfonamide
1-[1-(4-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]-4-(pyridin-4-yl)piperazine
4-[6-fluoro-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carbonyl]-1,3-dimethylpiperazin-2-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)pyrrolidin-3-yl]acetamide
1-(2-chloroprop-2-en-1-yl)-3-({methyl[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]amino}methyl)-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
N-(2-methoxyethyl)-1-[1-(2-phenoxypropanoyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
3-[3-({[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]amino}methyl)-1H-indol-1-yl]propanamide
2-(2-{[4-(1-methyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-pyrrol-1-yl)-1,3-thiazole
5-{[(1-hydroxy-2-methylpropan-2-yl)amino]methyl}-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-[(3S,4R)-1-(6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
2-[(4-chlorophenyl)methyl]-8-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,8-diazaspiro[4.5]decan-3-one
1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-cyclopropyl-2-(2-methoxyphenyl)pyridine-3-carboxamide
1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-4-(2-methoxybenzoyl)piperazine
N-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(2-methoxyphenoxy)piperidine
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(3-fluorophenoxy)ethan-1-one
7-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-1,3-diazepane-2,4-dione
8-[2-(benzenesulfonyl)ethyl]-2-butyl-2,8-diazaspiro[5.5]undecan-3-one
N,2-dimethyl-N-[1-(1,3-thiazol-2-yl)ethyl]-2-(thiophen-2-ylformamido)propanamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1H-pyrazole-3-carboxamide
N-[2-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy)propyl]-2,3-dimethyl-1H-indole-7-carboxamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-3-(pyrrolidine-1-sulfonyl)thiophene-2-carboxamide
(3S,9aR)-3-(cyclohexylmethyl)-8-[(1-phenyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(4-methoxyphenyl)-4-[1-(thiophen-3-ylmethyl)piperidin-3-yl]piperazine
5-(4-methyl-1,4-diazepan-1-yl)-2-({6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-2,3-dihydropyridazin-3-one
(1S,5R)-3-[3-(1H-pyrazol-1-yl)propanoyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2,5-dimethoxyphenyl)-N'-[2-(2-ethoxyphenyl)ethyl]propanediamide
1-({4-[3-(azepan-1-yl)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)azetidin-3-ol
2-[4-(2-amino-6-methoxypyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(1-propyl-1H-pyrazol-5-yl)acetamide
2,7-dimethyl-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-{[3-(2-fluorophenyl)-1H-pyrazol-5-yl]formamido}-3-phenylpropanoic acid
4-cyclopropyl-6-[4-(thian-4-yl)piperazin-1-yl]pyrimidine
8-(2,2-dimethylpropyl)-1-methyl-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-(2,3-dihydro-1H-inden-1-yl)-N-methylacetamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[(4-hydroxyquinolin-2-yl)methyl]piperidin-4-yl}propanamide
3-benzyl-8-(2,3-dihydro-1H-inden-2-yl)-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-fluorophenyl)-N-{[1-(1H-imidazol-4-ylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}acetamide
2-{[1-(2,6-dimethylpyrimidine-4-carbonyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
2-[(1S,5R)-6-[2-(2-chlorophenyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
4-chloro-1-methyl-3-{[3-(1H-pyrazol-5-yl)piperidin-1-yl]methyl}-1H-indazole
6-cyano-N-[(3R,5S)-5-(diethylcarbamoyl)-1-propanoylpyrrolidin-3-yl]pyridine-3-carboxamide
2-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-phenyl-1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidin-3-amine
N-methyl-2-(pyridin-3-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]pyrrolidin-3-yl]methanol
2-(dimethylamino)-N-ethyl-2-(4-fluorophenyl)-N-(2-methoxyethyl)acetamide