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2-({[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}amino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[3-(2-hydroxyethyl)-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-1-yl]-6-methylpyridine-3-carbonitrile
3-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
2-methoxy-5-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)pyridine
[1-(2-chlorophenyl)-2-(4H-1,2,4-triazol-4-yl)ethyl]dimethylamine
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
1-(6-hydroxy-1,4-oxazepan-4-yl)-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
methyl (2S,4S)-4-[2-chloro-5-(trifluoromethyl)benzamido]-1-[(3,5-dimethoxyphenyl)methyl]pyrrolidine-2-carboxylate
(3aS,7aR)-2-[(1-ethyl-1H-indol-4-yl)methyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2,7,8-trimethylquinoline-4-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1,3-thiazol-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-3,5-dimethyl-1H-pyrazole-4-sulfonamide
1-[2-(1H-indazol-5-yl)phenyl]ethan-1-one
8-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
1-{2-methoxy-4-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]phenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
1-[1-(2-aminoacetyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
4-[(2-methylpyridin-3-yl)oxy]-1-(1,3-thiazole-4-carbonyl)piperidine-4-carboxylic acid
methyl 3-[2-(methylsulfanyl)benzoyl]-7-oxo-9-(pyridin-4-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-N'-[2-(methylsulfanyl)phenyl]butanediamide
2-(2-hydroxyethyl)-9-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(1,3-dimethyl-4-phenyl-1H-pyrazol-5-yl)pyrrolidine-1-carboxamide
5-(6-aminopyridin-3-yl)-4-(4-methylphenyl)-N-[2-(morpholin-4-yl)ethyl]pyrimidin-2-amine
(1S,5R)-6-(2-methyl-1,3-thiazole-4-carbonyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-2-one
6-cyclopropyl-N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)pyrimidin-4-amine
3-(5-{[3-(methylsulfanyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)-1-(pyrrolidin-1-yl)propan-1-one
N-[2-(4-ethylmorpholin-2-yl)ethyl]-4,6-dimethyl-2-oxo-2H-pyran-5-carboxamide
methyl 8-[(2-methoxyphenyl)methyl]-1-(naphthalen-2-ylmethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
3-(1-methyl-1H-imidazol-2-yl)-1-(1-phenylcyclohexanecarbonyl)piperidine
3-[(2R,3R,6R)-5-(6-aminopyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
1-{2-oxo-2-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]ethyl}-1,2-dihydropyridin-2-one
methyl (2S,3S)-3-methyl-2-[(4-oxo-3,4-dihydroquinazolin-2-yl)formamido]pentanoate
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]-1-methyl-1H-pyrazole-3-carboxamide
2-[4-(4-ethyl-5-methylpyrimidin-2-yl)-1-[(4-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
[1-(3-fluorophenyl)propan-2-yl][(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]amine
(3R,4S)-4-cyclopropyl-1-[6-(4-fluorophenyl)pyridazin-3-yl]pyrrolidin-3-amine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-methylpyrrolidin-3-yl]-6-fluoro-4-hydroxyquinoline-3-carboxamide
N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-6-(propan-2-yl)-1H-indole-2-carboxamide
[(2,2-dimethyloxan-4-yl)methyl](methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-{5-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
2-[(4aS,8aR)-1-(2-methylpropyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-1,3-thiazole-4-carboxamide
N-[3-({[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]carbamoyl}amino)-4-methoxyphenyl]acetamide
2-{4-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}acetamide
3-{2-[3-(ethoxymethyl)-4-methoxyphenyl]-1H-imidazol-1-yl}pyridine
5-benzyl-4-{1-[(5-chlorothiophen-2-yl)sulfonyl]piperidin-4-yl}-2-methylpyrimidine
methyl 3-cyclobutanecarbonyl-7-oxo-9-[3-(pyridin-4-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
6-(4-methoxyphenyl)-9-(1-methyl-1H-pyrazole-5-carbonyl)-6,9-diazaspiro[4.5]decan-7-one
2-[3-methyl-4-({4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}methyl)-1H-pyrazol-1-yl]ethan-1-ol
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyridin-2-ylmethyl)acetamide