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N-ethyl-N-[2-(4-methylbenzenesulfonyl)ethyl]oxane-2-carboxamide
N-[(4-methoxypyridin-2-yl)methyl]-2-(pyridin-2-ylsulfanyl)acetamide
N-benzyl-3-({1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}oxy)benzamide
2-{[4-(4-cyclopentylpyrimidin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}[1-(dimethyl-1,3-thiazol-4-yl)ethyl]methylamine
3-chloro-4-({1-[2-(dimethylamino)acetyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
2-methyl-N-[2-(3-phenylpiperidin-1-yl)ethyl]-1-benzofuran-5-carboxamide
methyl 2-(diethylsulfamoyl)-6-[(4-methoxy-3-methylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}-N-(2-propylphenyl)piperazine-1-carboxamide
4-[4-(1-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]piperidine
1-(5-chloropyridin-2-yl)-4-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperazine
3-[4-(3-methylphenyl)piperazin-1-yl]-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]propanamide
5-(dimethylamino)-2-{2-[3-(morpholine-4-carbonyl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
[7-(4-methylpyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
1-[2-(diethylamino)ethyl]-4-(1H-pyrrole-3-carbonyl)-1,4-diazepan-6-ol
(4aS,7aR)-1-(1,2-oxazole-3-carbonyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]pyridin-2-amine
N-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
N-methyl-4-(propan-2-yl)-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyrimidin-2-amine
2-chloro-N-methyl-5-[(1E)-pent-1-en-1-yl]benzamide
5-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-N-methylpyrimidin-2-amine
N,1-dimethyl-N-[(4-phenoxyphenyl)methyl]-1H-pyrazole-3-carboxamide
methyl (1R,3S,3aR,6aS)-3-(2-fluoro-4-methylphenyl)-4,6-dioxo-5-phenyl-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N4,N4,5-trimethyl-N2-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]pyrimidine-2,4-diamine
2-{1-[(6-methylpyridin-2-yl)methyl]-4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperazin-2-yl}ethan-1-ol
4-(1-methyl-1H-1,2,4-triazol-5-yl)-2-{octahydropyrrolo[1,2-a]piperazin-2-yl}pyrimidine
[2-(2-methyl-1H-indol-1-yl)ethyl][1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
N-cyclopentyl-4,4,4-trifluoro-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)butanamide
(3S,4S)-1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]acetamide
N-{[1-(2-fluorophenyl)cyclopentyl]methyl}-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N2,N2,5,6-tetramethyl-N4-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]pyrimidine-2,4-diamine
ethyl 1-(4-methoxyphenyl)-5-[({[1-(morpholin-4-yl)cyclopentyl]methyl}amino)methyl]-1H-pyrazole-4-carboxylate
N-[(3S,4R)-4-hydroxyoxolan-3-yl]-N-methyl-3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)benzene-1-sulfonamide
4-methoxy-6-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]pyrimidin-2-amine
N-[(3,4-difluorophenyl)methyl]-3-{1-[2-(phenylsulfanyl)acetyl]piperidin-3-yl}propanamide
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-2-(1H-pyrazol-1-yl)butanamide
2-(3-fluoro-4-hydroxyphenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
2-(cyclopentylmethyl)-1-(2-methoxyethyl)-3-[4-(3-methoxyphenyl)piperazine-1-carbonyl]-6-methyl-1,4-dihydropyridin-4-one
4-(5-{[4-(oxolan-2-ylmethyl)piperazin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoic acid
6-ethyl-5-methyl-N4-[3-(4H-1,2,4-triazol-4-yl)propyl]pyrimidine-2,4-diamine
1-[2-methyl-4-({3-[(pyridin-3-yl)amino]propyl}amino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
(2E)-N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-3-(1H-imidazol-4-yl)prop-2-enamide
N,N-dimethyl-1-(6-methyl-2-propylpyrimidin-4-yl)pyrrolidin-3-amine
3-[5-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
1-[1-(benzyloxy)-2-oxo-1,8-diazaspiro[4.5]decan-8-yl]-4-phenylbutane-1,4-dione
(1S,5R)-3-{[3-(3-methoxyphenyl)phenyl]methyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(cyclohexylamino)-1-(2-phenylethyl)pyrrolidin-2-one
3-{[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-5-(2-methylpropyl)-1H-pyrazole
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-2-[3-(2-fluorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide