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2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-[3-(2-phenylethyl)piperidin-1-yl]ethan-1-one
N,7-dimethyl-N-(thiophen-3-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
[1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-2-yl]methanol
methyl 2-[4-({[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]carbamoyl}amino)phenoxy]acetate
1-(2-ethoxyethyl)-N-[2-(1H-imidazol-1-yl)ethyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-methyl-4-(3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}phenyl)butan-2-ol
6-methyl-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]pyridine-2-carboxamide
2-{1-[(1-cycloheptanecarbonylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}-2-(1,3-thiazol-2-yl)piperidine-1-carboxamide
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,1-benzoxazole-3-carboxamide
N3-[(2-fluorophenyl)methyl]-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-[(4-{2-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl]piperazine-1-carbaldehyde
(2S,4R)-4-amino-1-[2-(3-cyano-2-methyl-1H-indol-1-yl)acetyl]-N,N-diethylpyrrolidine-2-carboxamide
2-methoxy-N-{4-[3-(1H-pyrazol-3-yl)phenyl]phenyl}acetamide
(2R)-2-methyl-1-[3-(1H-1,2,4-triazol-3-yl)benzoyl]piperazine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methylpyridine-4-carboxamide
(4R)-4-(1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane-6-carbonyl)-1,3-thiazolidin-2-one
9-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]-7-(5-methylthiophen-2-yl)-4-(pyridine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]thiophene-3-sulfonamide
(3S,4R)-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
2-amino-4-(2H-1,3-benzodioxol-5-yl)-6-(3,5-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
1-(cyclopropylmethyl)-5-[(2,6-difluorophenyl)methyl]-N-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-{[1-(2H-1,3-benzodioxol-5-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
N-[(2S)-1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-1-oxopropan-2-yl]acetamide
5-(2-chloro-4-fluorophenyl)pyridine-2-carbonitrile
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
1-[1-(5-methyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidine
3-(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}thiophen-3-yl)prop-2-yn-1-ol
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-(1H-pyrazol-4-yl)pyridine-3-carboxamide
5-(2,3-dimethylquinoxaline-6-carbonyl)-N-(3-methoxypropyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
6-(piperidin-3-yl)-N-(prop-2-en-1-yl)-N-(pyridin-3-ylmethyl)pyrimidin-4-amine
N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-4-ylmethyl)oxane-2-carboxamide
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(but-3-enoyl)piperidine-4-carboxamide
methyl 6-[(2,4-dimethylphenyl)methyl]-2-(thiomorpholine-4-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(3-methoxyphenyl)methyl]-3-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-3-yl]propanamide
dimethyl[1-(3-{1-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]-4-phenyl-1H-imidazol-5-yl}phenyl)ethyl]amine
3-(4-fluorophenyl)-N-[(1r,4r)-4-methoxycyclohexyl]benzamide
4-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-1,4-diazepan-2-one
3-(2-phenylethyl)-8-[2-(1H-1,2,4-triazol-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-ol
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(2,3-dimethylphenyl)methyl]pyrimidin-2-amine
1-ethyl-N-{[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]methyl}-5-oxopyrrolidine-3-carboxamide
(4aS,8aS)-2-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-decahydroisoquinolin-4a-ol
3-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-2,8-diazaspiro[4.5]decane
5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-1H-indole
N-methyl-N-(oxolan-3-yl)-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide