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N-{2-methyl-2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-5-(1-methylpyrrolidin-2-yl)thiophene-2-carboxamide
N-(4-cyano-2-ethylphenyl)-3-[(3-oxopiperazin-1-yl)methyl]benzamide
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(2-phenoxyethyl)piperazine
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(4-hydroxyphenyl)ethan-1-one
(3aR,6aS)-5-{[3-methoxy-4-(prop-2-en-1-yloxy)phenyl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{[5-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]methyl}pyridine
1-[2-({ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
(2E)-1-{7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(pyridin-3-yl)prop-2-en-1-one
N-[1-(4-hydroxyphenyl)-2-methylpropan-2-yl]-4-(1H-pyrazol-4-yl)butanamide
2-[(2-carbamoylmorpholin-4-yl)methyl]benzoic acid
1-{2-[2-(1-phenyl-1H-pyrazol-5-yl)-1H-imidazol-1-yl]ethyl}pyrrolidin-2-one
N-cyclohexyl-3-[(3R)-3-fluoropyrrolidin-1-yl]propanamide
N-{[1-(1H-1,3-benzodiazol-2-ylmethyl)pyrrolidin-3-yl]methyl}-1H-pyrrole-2-carboxamide
3-[(3-hydroxypiperidin-3-yl)methyl]-1-[4-(4-methoxyphenoxy)phenyl]urea
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1-[1-(2-methoxyphenyl)propan-2-yl]-1-methyl-3-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}urea
(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-7-{[(4-methylphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-{4-[(ethylcarbamoyl)amino]-3-methoxyphenyl}-2-(morpholin-4-yl)acetic acid
N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]-2,1-benzoxazole-3-carboxamide
4-(1-{1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}ethyl)morpholine
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
5-chloro-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
3-[(2R)-2-methylpiperazine-1-carbonyl]-N-(oxan-4-ylmethyl)benzene-1-sulfonamide
(1S,5R)-6-(cyclobutylmethyl)-3-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
6-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]quinoxaline
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
(3aS,6aR)-5-{furo[3,2-c]pyridin-4-yl}-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-{1-cyclohexyl-3-[(2-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}-3,4-dihydropyrimidin-4-one
4,6-dimethyl-2-oxo-N-[(1R)-2,2,2-trifluoro-1-phenylethyl]-1,2-dihydropyridine-3-carboxamide
4-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-6-methoxypyrimidine
3-hydroxy-1-methyl-3-({methyl[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)piperidin-2-one
4-[3-(furan-2-yl)phenyl]-1-[2-(1H-imidazol-4-yl)ethyl]-1H-1,2,3-triazole
1-methyl-4-{1-[1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}piperazine
2-phenyl-1-[1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]ethan-1-ol
2-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-4-carbonitrile
2-[methyl({4-methyl-5-[1-(1H-pyrrole-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N-methyl-2-(4-phenylpiperidin-1-yl)acetamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-phenylbutanamide
{2,4,6-trimethyl-3-[({[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amino)methyl]phenyl}methanol
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-(9H-purin-6-yl)piperidin-4-amine
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-2-(thiophen-3-yl)acetamide
(2S,4S)-N,N-diethyl-4-(2-hydroxyacetamido)-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}pyrrolidine-2-carboxamide
1-(carbamoylmethyl)-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methylpiperidine-3-carboxamide
N-[2-(1H-imidazol-1-yl)ethyl]-N-methyl-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
4-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}morpholine-2-carboxamide
N-[2-(1-benzylpyrrolidin-3-yl)ethyl]-1,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(4-ethoxyphenyl)methyl]-N-(2-methoxyethyl)-1-(propan-2-yl)pyrrolidine-3-carboxamide
N-{1-[7-(furan-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}pyridine-3-carboxamide
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-4-methyl-N-(pyridin-4-ylmethyl)-1,2,5-oxadiazole-3-carboxamide