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N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(pyrrolidin-1-yl)pyrimidine-5-carboxamide
1-[3-(1H-imidazol-2-yl)benzoyl]-4-(3-methoxybenzoyl)piperazine
N-[(2-fluorophenyl)methyl]-3-{1-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]piperidin-3-yl}propanamide
4-[5-cyclopropyl-3-(phenoxymethyl)-1H-1,2,4-triazol-1-yl]benzene-1-sulfonamide
(2R,6R)-4-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-methyl-2-(2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamido)acetamide
5-(2-chloro-4-fluorophenoxymethyl)-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-1,2-oxazole-3-carboxamide
2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,N,5-trimethylpyrimidin-4-amine
methyl 4-({4-[2-(2-fluorophenyl)-1-[N-methyl-1-(2-methylfuran-3-yl)formamido]ethyl]piperidin-1-yl}methyl)benzoate
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-methyl-1-[3-(piperidin-1-ylmethyl)phenyl]urea
2-[2-chloro-4-({cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]acetamide
(3S,5R)-1-(4-hydroxy-3-methylbenzoyl)-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
3-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-1-[2-(2-methoxyethoxy)phenyl]urea
(2R,6R)-4-[(1r,4r)-4-methylcyclohexanecarbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-[3-benzyl-3-(hydroxymethyl)piperidin-1-yl]pyridine-4-carboxamide
6-tert-butyl-N-methyl-2-oxo-N-(quinolin-4-ylmethyl)-2,3-dihydropyrimidine-4-carboxamide
1-[(3S)-3-ethylmorpholin-4-yl]-4-(1H-imidazol-1-yl)butan-1-one
N,N-dimethyl-7-(2-methylbenzenesulfonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-5-phenyl-1,2-oxazole-3-carboxamide
2-methoxy-N-{1-[1-(3-methoxypropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
(2R,3R,6R)-3-(4-methylphenyl)-5-(4-methylpyrimidine-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,2,7,8-tetramethylquinoline-4-carboxamide
4-(4-methylpentanoyl)-N-[2-(methylsulfanyl)phenyl]morpholine-2-carboxamide
N-[3-(2-methoxyethoxy)phenyl]-3-(2-methylpiperidin-1-yl)azetidine-1-carboxamide
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-1-[(3-hydroxy-4-methoxyphenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-[2-(3-fluorophenyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{2-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
1-(dimethyl-1,3-oxazole-4-carbonyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
ethyl 4-[2-(pyridin-4-yl)pyrimidine-5-amido]piperidine-1-carboxylate
(3aS,7aR)-5-methyl-2-[4-(1H-pyrazol-4-yl)butanoyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
4-[1-ethyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]-2,6-dimethylpyrimidine
2-amino-6-(2,2-dimethyloxan-4-yl)-4-(2-ethylpyrimidin-5-yl)-5-propylpyridine-3-carbonitrile
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-phenylethane-1,2-dione
4-[3-(5-methylthiophen-2-yl)-5-(thiomorpholine-4-carbonyl)benzenesulfonyl]morpholine
N'-cyclopentyl-N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]butanediamide
2-(3-{[(2-methoxyethyl)(1-methylpiperidin-4-yl)amino]methyl}phenyl)-6-methyl-3,4-dihydropyrimidin-4-one
N-{3-[2-(4-hydroxypiperidin-1-yl)acetamido]phenyl}-3-phenylpropanamide
(2,1,3-benzoxadiazol-4-ylmethyl)[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]methylamine
4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-1-(furan-2-ylmethyl)piperidine
{[2-(furan-2-yl)pyrimidin-5-yl]methyl}(methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(5-methylthiophene-2-carbonyl)piperidine
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(pyridin-2-ylsulfanyl)acetamide
1-methanesulfonyl-4-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-1,4-diazepane
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}[1-(2-methoxyphenyl)ethyl]methylamine
2-ethoxy-4-({4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)phenol
N-[(3S,7S,8aS)-1,4-dioxo-3-propyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,5-dichlorobenzamide
1-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one