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4-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]benzene-1-sulfonamide
3-{5-[(4-chloro-3-fluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
6-methyl-2-(piperidin-1-yl)-N-(piperidin-3-ylmethyl)pyrimidin-4-amine
5-chloro-N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}thiophene-2-carboxamide
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
4-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-N,N-dimethyl-4-oxobutanamide
(3S,9aR)-3-[(benzyloxy)methyl]-8-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(4-chlorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]ethan-1-one
(3S,4S)-3-{[(5-tert-butyl-1H-pyrazol-3-yl)methyl](methyl)amino}-4-hydroxy-1λ6-thiolane-1,1-dione
2-{4-[(dimethylamino)methyl]phenyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-({[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)-N-(1-methyl-1H-1,2,4-triazol-3-yl)benzamide
4-[(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)methyl]benzamide
1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butane-1,2-dione
2-(1H-1,3-benzodiazol-1-yl)-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]acetamide
5-methyl-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
3-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}-N-[5-(trifluoromethyl)-1,3,4-oxadiazol-2-yl]benzamide
2-{4-[1-(3,5-dimethylphenyl)piperidin-4-yl]piperazin-1-yl}pyrimidine
4-ethyl-5-methyl-N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]pyrimidin-2-amine
{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
N-ethyl-5-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]pyrimidin-2-amine
3-(3,4-dimethylphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]propan-1-one
3-[(4-methoxyphenyl)methyl]-1-methyl-8-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[3-(4-ethylpiperazine-1-carbonyl)-1,2-oxazol-5-yl]methyl}(methyl)(2-phenylethyl)amine
6-[1-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]pyrimidin-4-ol
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
N-[(5-chloro-2-ethoxyphenyl)methyl]-N-methyl-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
[(2-fluorophenyl)methyl][(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl](2-methoxyethyl)amine
1-(2,2-diphenylethyl)-4-(hydroxymethyl)piperidin-4-ol
N-[1-(3-methoxypyrazin-2-yl)piperidin-4-yl]methanesulfonamide
N-[2-(4-fluorobenzenesulfonyl)ethyl]-2,6-dimethylpyridine-4-carboxamide
2-methyl-N-{1-[1-(3-phenylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
2-methoxy-1-{4-[(2-methylphenyl)methyl]piperazin-1-yl}ethan-1-one
1-[cyclopropyl(4-methylpyridin-2-yl)methyl]-3-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)urea
N-(2-methoxyethyl)-3-(1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)propanamide
6-{[(3R,4S)-1-(1-acetylpiperidin-4-yl)-4-propylpyrrolidin-3-yl]amino}pyridine-3-carbonitrile
3-(1-{1-[(2R)-2-aminopropanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-chlorophenyl)urea
8-(4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}-1-(2-methoxyphenyl)-1H-1,2,4-triazole
N-(2-methoxyphenyl)-3-(4-phenylbenzoyl)piperidine-1-carboxamide
(4aR,7aS)-4-[(3,5-difluorophenyl)methyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(4aS,7aR)-1-(5-methyl-1,3-oxazole-4-carbonyl)-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(5-methylthiophene-2-carbonyl)piperidine
4-({4-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]piperazin-1-yl}methyl)benzene-1,2-diol
2-[N-(3-fluorophenyl)methanesulfonamido]-N-[2-(1H-imidazol-4-yl)ethyl]acetamide
2-amino-N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carboxamide
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
2-{4-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
N-(1-hydroxybutan-2-yl)-2-(methylsulfanyl)-N-(thiophen-2-ylmethyl)pyridine-3-carboxamide