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(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(2-fluorobenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3R,4R)-3-cyclobutyl-1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-4-methylpyrrolidin-3-ol
4-chloro-N-[2-(dimethylamino)-2-(4-methylphenyl)ethyl]-1-methyl-1H-pyrazole-3-carboxamide
5-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-N-ethylpyrimidin-2-amine
1-{[3-(methylsulfanyl)phenyl]methyl}-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-4-carboxamide
5-cyclopropanecarbonyl-1'-(5-methylpyrazine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{[4-(1,2-oxazolidine-2-carbonyl)-1,3-oxazol-2-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
3-{[(1-methyl-1H-imidazol-2-yl)methyl](propyl)amino}-1-(3-methylpiperidin-1-yl)propan-1-one
2,6-dimethyl-5-{2-oxo-2-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
1-{[1-(6-{[(2-methylphenyl)methyl]amino}pyridine-3-carbonyl)piperidin-4-yl]methyl}pyrrolidin-2-one
2-amino-4-methyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1,3-thiazole-5-carboxamide
N-[2-(diethylamino)ethyl]-N-methyl-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
N-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-4-(5-methyl-4H-1,2,4-triazol-3-yl)aniline
6-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-cyclopropyl-1-[2-(dimethylamino)ethyl]-6-methyl-4-oxo-2-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
5-({spiro[azepane-4,2'-chromene]-1-yl}carbonyl)-1H-1,2,4-triazol-3-amine
(3S,4R)-4-methyl-1-[5-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-3-carbonyl]piperidine-3,4-diol
1-methyl-2-{1-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}-1H-1,3-benzodiazole
5-(2-chlorophenyl)-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}furan-2-carboxamide
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(2,2-diphenylethyl)propanamide
4-[3-(1-methoxyethyl)phenyl]-5-(methoxymethyl)-3-methyl-1H-pyrazole
1-[2-(2-methoxyethyl)piperidin-1-yl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
2,5-dimethyl-3-{4-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl}pyrazine
3-{methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}-1-phenylpropan-1-ol
8-fluoro-2-{[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]methyl}-1,4-dihydroquinolin-4-one
4-[(2-aminopyridin-3-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(1H-imidazol-1-yl)-1-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butan-1-one
2-acetamido-N-[(4-methoxyphenyl)methyl]-N-(2-methylpropyl)acetamide
3-methyl-1-{1-[6-(3,3,4-trimethylpiperazin-1-yl)pyridine-3-carbonyl]piperidin-3-yl}butan-1-one
3-{[4-(benzyloxy)piperidin-1-yl]methyl}piperidin-3-ol
N-[1-(hydroxymethyl)cyclopentyl]-4-(quinolin-6-yloxy)piperidine-4-carboxamide
7-(3-methoxypropyl)-2-{2-[methyl(phenyl)amino]acetyl}-2,7-diazaspiro[4.5]decan-6-one
2-({[(3R,4R)-4-(hydroxymethyl)-1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-(furan-2-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
N-[(3R,4S)-1-benzoyl-4-cyclopropylpyrrolidin-3-yl]-2-(methylamino)-1,3-thiazole-4-carboxamide
3-(1-methyl-6-oxopiperidin-3-yl)-1-(2-propylphenyl)urea
3-[3-methyl-1-(2-methylphenyl)-1H-pyrazol-5-yl]-1-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}urea
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-{3-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
2,4-dichloro-3-{[4-(oxolane-2-carbonyl)-1,4-diazepan-1-yl]methyl}phenol
N-cyclopropyl-N-[(5-methylthiophen-2-yl)methyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-{1-[(3-methylphenyl)methyl]cyclopropyl}-3-(1-methylpiperidin-3-yl)propanamide
4-{3-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}morpholine
4-{2-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-1-yl}phenol
2-[(2-{[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)methyl]carbamoyl}phenyl)amino]acetic acid
2-(3,3-diphenylpiperidine-1-carbonyl)-6-methyl-4H-pyran-4-one
3-cyclopropyl-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-1H-pyrazole-5-carboxamide
3-(1-benzofuran-2-yl)pyrazine-2-carbonitrile