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1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
5-methanesulfonyl-2-methyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}pyrimidin-4-amine
2-amino-6-(4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)-3,4-dihydropyrimidin-4-one
{3-[(3-chlorophenyl)methyl]-1-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]piperidin-3-yl}methanol
2-(2-fluoro-4-methoxyphenyl)-5-methyl-4-[(4-methyl-1H-pyrazol-1-yl)methyl]-1,3-oxazole
5-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}-1-(2-phenylethyl)-1H-1,2,4-triazole
2-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidine-1-carbonyl}phenol
N-methyl-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
1-methyl-N-(2-phenylethyl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidin-4-amine
N-ethyl-N-(4-hydroxybutyl)-2-methyl-1-benzofuran-5-carboxamide
4-(2,4-dioxoimidazolidin-1-yl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]benzamide
3-(1,3-benzothiazol-2-yl)-1-(thiomorpholin-4-yl)propan-1-one
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}acetamide
1-(1-{3-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}piperidin-3-yl)propan-1-one
4-benzyl-7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
3-fluoro-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
1-{3-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}azepan-2-one
5-{5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazol-1-yl}pentan-1-amine
7-(2,3,4,9-tetrahydro-1H-carbazole-1-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-chloro-N-[1-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
(1S,5R)-6-benzyl-3-(1H-imidazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(3-fluorophenyl)methyl]-4-[(1-propylpiperidin-4-yl)amino]pyrrolidin-2-one
1-{[4-(2-hydroxyethoxy)phenyl]methyl}-4-methylpiperidine-4-carbonitrile
methyl 5-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-(furan-2-ylmethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-chloro-N-ethyl-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(oxolan-2-ylmethyl)benzamide
9-{[3-(methylsulfanyl)phenyl]methyl}-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-({4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-2,6-dimethylphenol
2-[(1S,5R)-3-[(3,4-dimethoxypyridin-2-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
1-[4-(3-chloro-4-fluorophenyl)piperazin-1-yl]-3-(1-methyl-1H-pyrazol-5-yl)propan-1-one
1-methyl-N-(2-phenylethyl)-N-(1,3-thiazol-4-ylmethyl)piperidin-4-amine
(2-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)urea
2-methoxy-1-[4-(3-phenylbutyl)-1,4-diazepan-1-yl]ethan-1-one
N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}-2-methylpropanamide
dimethyl(3-{2-[2-(2-methylphenyl)pyrimidin-5-yl]-1H-imidazol-1-yl}propyl)amine
N-(1-carbamoylcycloheptyl)-7-methyl-1-benzofuran-2-carboxamide
5-phenyl-3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}-1,2,4-triazine
7-(1,3-benzothiazol-2-yl)-4-(5-methylpyridine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-{[3-(morpholin-4-yl)phenyl]methyl}-decahydro-2,7-naphthyridine-2-carboxamide
N-benzyl-2-(2-oxo-1,2,3,4-tetrahydroquinolin-1-yl)-N-(oxolan-2-ylmethyl)acetamide
4-amino-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}butanamide
1-(4-fluorophenyl)-4-[4-(2-methylpyrimidin-4-yl)piperidin-1-yl]butane-1,4-dione
(3S,4S)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
(3R,4R)-1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
4-[(dimethylamino)methyl]-1-[(4-fluorophenyl)methanesulfonyl]azepan-4-ol
4-[(5-methylfuran-2-yl)methyl]-3-{2-oxo-2-[4-(pyrazin-2-yl)piperazin-1-yl]ethyl}piperazin-2-one
[(3R,4R)-1-[(2-chloro-3,4-dimethoxyphenyl)methyl]-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
N-{[3-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)-1,2,5-thiadiazole-3-carboxamide
(3R,9aR)-3-benzyl-8-[(4-chlorophenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione