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4,6-dimethyl-N-[1-(3-phenylpropyl)piperidin-3-yl]pyrimidin-2-amine
3-(methoxymethyl)-1-[(6-methoxynaphthalen-2-yl)methyl]pyrrolidine
2-(2-{[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
3-hydroxy-1-[(3-methylphenyl)methyl]-3-({[(3-methylpyridin-2-yl)methyl]amino}methyl)piperidin-2-one
5-{[(2-hydroxyethyl)({[4-(methylsulfanyl)phenyl]methyl})amino]methyl}-2-methoxyphenol
3-methyl-N-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)-1,2-oxazole-5-carboxamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-ethoxyacetamide
5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}quinoxaline
1-(1,4-dithiepan-6-yl)-3-[4-(methylsulfanyl)benzoyl]piperidine
N-(2-methoxyethyl)-1-{1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidin-4-yl}piperidine-3-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-({4-[1-(2,3-dihydro-1H-inden-2-yl)-3-methyl-1H-1,2,4-triazol-5-yl]-1H-1,2,3-triazol-1-yl}methyl)piperidine
2-ethyl-9-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
1-{[2-(butan-2-ylsulfanyl)pyrimidin-5-yl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
2-(5-ethyl-1-benzofuran-3-yl)-1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
1-(azocan-1-yl)-3-(2-methoxy-4-{[(2-phenoxyethyl)amino]methyl}phenoxy)propan-2-ol
6-chloro-3-({ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-N,N-dimethylimidazo[1,2-a]pyridine-2-carboxamide
2-[(3,4-dimethoxyphenyl)methyl]-N-[2-(methylsulfanyl)ethyl]-1,3-benzoxazole-6-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[(3R,4S)-4-(5-methylfuran-2-yl)-1-(propan-2-yl)pyrrolidin-3-yl]morpholine-4-sulfonamide
7-(cyclopropylmethyl)-2-methyl-N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-{[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]amino}-N,5-dimethyl-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)piperidin-2-one
4-phenyl-N-({1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-3-yl}methyl)benzamide
1-[3-(2-phenylethyl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
(2S,4R)-1-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-4-amino-N-ethylpyrrolidine-2-carboxamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(thiophen-3-ylmethyl)pyrrolidine-3-carboxylic acid
N-[1-(cyclopropylmethyl)-1H-indazol-3-yl]-2-[3,5-dimethyl-4-(pyridin-4-yl)-1H-pyrazol-1-yl]acetamide
1-(2-ethoxyethyl)-N-methyl-2-oxo-N-(pyridin-2-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-(1H-imidazol-2-ylmethyl)-N-methyl-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
3-fluoro-2-methoxy-N-{[1-(oxan-4-yl)pyrrolidin-3-yl]methyl}benzamide
N-(2,3-dimethylphenyl)-N'-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}ethanediamide
(3S,4S)-4-propyl-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidine-3-carboxylic acid
3-(2H-1,3-benzodioxol-5-yl)-5-(4,4,4-trifluorobutan-2-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
5-oxo-1-[3-(propan-2-yloxy)propyl]pyrrolidine-3-carboxylic acid
1-[(3-methoxyphenyl)methyl]-3-(5-methylfuran-2-yl)-5-(oxolan-3-yl)-1H-1,2,4-triazole
methyl 2-{4-[(4-methyl-1,3-thiazol-5-yl)methyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl}acetate
2-ethyl-4-phenyl-9-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-2,9-diazaspiro[5.5]undecane
(3R,4R)-1-[2-chloro-5-(piperidin-1-yl)benzoyl]-4-ethylpiperidine-3,4-diol
5-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-4-yl}-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1H-imidazol-2-ylmethyl)-N-methylacetamide
N-[3-(4-methylpiperazin-1-yl)propyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
2-{4-[3-(thiophen-3-yl)propyl]-1,4-diazepan-1-yl}-1,3-benzothiazole
6-(pyrrolidin-1-ylmethyl)-4-(1,3-thiazol-2-yl)-1,4-oxazepan-6-ol
2-tert-butyl-4-hydroxy-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)pyrimidine-5-carboxamide
5-(2,3-dihydro-1-benzofuran-7-carbonyl)-3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-[2-(cyclohex-1-en-1-yl)pyrimidin-4-yl]piperidin-3-ol
2-[(4aS,8aS)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-5,6-dimethylpyridine-3-carboxylic acid