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2-propanoyl-N-[2-(pyridin-2-yl)ethyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1,3-dimethyl-N-[(3-methyloxetan-3-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-benzyl-N3-[2-(cyclohex-1-en-1-yl)ethyl]-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-benzyl-3-ethyl-1-(6-oxo-1,6-dihydropyridazine-3-carbonyl)-1,4-diazepan-5-one
1-(2-methoxyphenyl)-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1H-pyrazole
4-{2-[(3-chlorophenyl)methyl]-1,3-benzoxazole-6-carbonyl}piperazin-2-one
methyl[(5-methylthiophen-2-yl)methyl]{[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
3-benzyl-1-(quinolin-2-yl)piperidine-3-carboxylic acid
3-{3-[2-(4-fluoro-3-methylphenyl)pyridin-4-yl]pyrrolidine-1-carbonyl}cyclobutan-1-one
3,6-dimethyl-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1-benzofuran-2-carboxamide
4-(3-chlorophenyl)-3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4H-1,2,4-triazole
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
2-(4-{[3-hydroxy-1-(2-methoxyethyl)-2-oxopiperidin-3-yl]methyl}piperazin-1-yl)pyridine-3-carbonitrile
2-(dimethylamino)-N-[5-({[(1S)-2-hydroxy-1-phenylethyl]carbamoyl}amino)-2-methylphenyl]acetamide
3-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
1-(4-fluorophenyl)-3-(2-methylpropyl)-5-(oxolan-3-yl)-1H-1,2,4-triazole
N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]-N'-phenylethanediamide
N-(1-{1-[(5-cyclohexylthiophen-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(quinolin-2-ylmethyl)pyrrolidin-3-yl]methanol
methyl (3aS,6aS)-2-(1-methanesulfonylpiperidin-4-yl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylate
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
5-{[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-3-methyl-1H-pyrazole
N-[(3R,4R)-3-hydroxy-1-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}piperidin-4-yl]pyridine-2-carboxamide
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(oxolan-2-ylmethyl)amine
N-methyl-3-{methyl[(2-methylquinolin-8-yl)carbamoyl]amino}butanamide
2-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}acetic acid
N-[(3S,4R)-1-[(1-methyl-1H-indol-2-yl)methyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
4-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-5,6,7,8-tetrahydroquinoline-3-carboxamide
7,7-dimethyl-2-[(2R)-oxolan-2-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-[4-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperazine-1-carbonyl]morpholine
[(3R,4R)-4-(azepan-1-ylmethyl)-1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanol
1-(pyridin-4-ylmethyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
5-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]pyridine-2-carbonitrile
N-benzyl-N-methyl-3-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
1-[3-(4-fluorophenyl)phenyl]-3-{[4-(hydroxymethyl)oxan-4-yl]methyl}-3-methylurea
3-[2-(2,6-difluorophenyl)ethyl]-1-(4-methyl-1,3-oxazole-5-carbonyl)piperidine
N-(2-hydroxyethyl)-N-methyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
2-cyclopentyl-1-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
1-(2-methoxyphenyl)-4-{1-[2-(methylsulfanyl)benzoyl]piperidin-3-yl}piperazine
1-[2-(piperazin-1-yl)ethyl]-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
7,11-dimethyl-3-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]-3,7,11-triazaspiro[5.6]dodecane
3-(6-methoxynaphthalene-2-carbonyl)piperidine
2-(furan-3-yl)-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridine
6-(methoxymethyl)-N-{2-[4-(propan-2-yl)-1,3-thiazol-2-yl]ethyl}pyrimidin-4-amine
[5-methyl-7-(2-methyl-5-propylpyrimidin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
N-[(3S,4R)-4-(4-methylphenyl)-1-[3-(methylsulfanyl)propanoyl]pyrrolidin-3-yl]acetamide
8-(2-methyl-1,3-thiazole-5-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
4-chloro-N-methyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-2-propanamidobenzamide
({4-ethyl-5-[1-(isoquinolin-1-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine