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5,5-dimethyl-3-{2-oxo-2-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl}-1,3-oxazolidine-2,4-dione
2-{3-[(3aS,6aS)-octahydropyrrolo[3,4-b]pyrrol-5-ylmethyl]phenoxy}acetamide
1-{2-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonane-7-carbonyl]phenyl}ethan-1-one
1-[4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-3-phenylpyrrolidin-3-ol
3-(1-methyl-1H-pyrazol-4-yl)-1-(3-{[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)propan-1-one
(1s,4s)-4-{[ethyl(oxan-4-ylmethyl)amino]methyl}cyclohexan-1-amine
3-butanamido-N-[(4-phenyloxan-4-yl)methyl]benzamide
2-[1-(3-methylbutyl)-4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperazin-2-yl]ethan-1-ol
2-{[benzyl(1,3-thiazol-2-ylmethyl)amino]methyl}benzoic acid
4-[(2,5-difluorophenyl)methyl]-9-methoxy-7-(4-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-butyl-5-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-1,3-benzoxazole
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}urea
ethyl 4-(3,6,7-trimethyl-1-benzofuran-2-amido)piperidine-1-carboxylate
3-ethyl-N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1H-indole-2-carboxamide
(2S,4R)-1-[(2-chloro-6-fluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-methyl-N-(1H-pyrazol-5-ylmethyl)pyrrolidine-2-carboxamide
(1S,5R)-3-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
5-chloro-2-methoxy-4-[3-(4H-1,2,4-triazol-4-yl)phenyl]pyridine
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
5-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-4-phenylbutane-1,4-dione
(3S,4S)-4-[methyl({3-[(4-methylphenyl)sulfanyl]propyl})amino]-1-[(4-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-ol
N-[(4-methoxyphenyl)methyl]-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
2-phenyl-7-[2-(1H-pyrazol-1-yl)butanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(4aS,7aR)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(4-fluorophenyl)-1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}piperidin-4-ol
5-[(4-acetyl-4-phenylpiperidin-1-yl)methyl]-2-methoxybenzoic acid
5-[3-(2-fluorophenoxymethyl)piperidine-1-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
1-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-4-(oxolan-3-yl)-1H-1,2,3-triazole
2-{1-[4-(2,4-difluorophenyl)-1H-1,2,3-triazol-1-yl]ethyl}-1H-1,3-benzodiazole
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-2,6-dimethylpyrimidine-4-carboxamide
2-(furan-2-yl)-2-oxo-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]acetamide
(2E)-3-(1-methyl-1H-pyrazol-4-yl)-1-[3-(naphthalene-1-carbonyl)piperidin-1-yl]prop-2-en-1-one
2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]benzonitrile
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
methyl (2S,4S)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(2,3-dimethoxyphenyl)methyl]pyrrolidine-2-carboxylate
2-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
4-methyl-3-[4-(pyridin-4-yl)piperidine-1-carbonyl]benzene-1-sulfonamide
8-(3-hydroxypropyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-{2-[4-(morpholin-4-ylmethyl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
2-(3-hydroxypropyl)-9-[2-(4-methylphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
ethyl[(4-methanesulfonylphenyl)methyl](oxan-4-ylmethyl)amine
N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(3,4-dimethylphenyl)ethan-1-one
3-cyclopropyl-5-(2,6-difluoro-3-methylphenyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-3-[6-(dimethylamino)-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]urea
2-benzyl-8-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]acetyl}-2,8-diazaspiro[4.5]decan-3-one
(3S,9aR)-8-(naphthalene-1-sulfonyl)-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-benzyl-1-[2-(pyrrolidin-3-yl)benzoyl]piperidin-4-ol
2-[4-(4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
(2S,4S)-4-amino-1-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide