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4-{[3-(dimethyl-1,3-thiazol-2-yl)phenyl]methyl}morpholine
N-(quinolin-2-ylmethyl)pyridazine-4-carboxamide
N-(butan-2-yl)-N-(pyridin-3-ylmethyl)-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
2-cyclopropyl-9-(3-methylbut-2-en-1-yl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-1-{1-[(3-methylphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
N-[(3S,4R)-4-hydroxyoxolan-3-yl]-N,3,4,7-tetramethyl-1H-indole-2-carboxamide
4-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)phenol
2-methyl-N-[2-(1H-1,2,3-triazol-1-yl)ethyl]-1,3-thiazole-4-carboxamide
3-[1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-1-(4-methylpiperazin-1-yl)propan-1-one
2-(3-fluorophenyl)-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidine
(2S,4R)-4-amino-N,N-diethyl-1-(2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}acetyl)pyrrolidine-2-carboxamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-4-propylpyrimidine-5-carboxamide
(9aR)-8-benzyl-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-(1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-2-methylpropan-2-yl)morpholine
N-[(2-methoxyphenyl)methyl]-2-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]acetamide
1-(4-ethylpiperazin-1-yl)-3-[3-({methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-[(2-methylpyrrolidin-1-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
5-methyl-N-[(3-methyloxetan-3-yl)methyl]-4-[(prop-2-en-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
3,5-dimethyl-N-(2-oxoazepan-3-yl)-1H-indole-2-carboxamide
4-(1-aminocyclobutanecarbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(1R,2R,6S,7S)-N-{4-[2-(pyridin-2-yl)ethoxy]phenyl}-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
5-(benzenesulfonyl)-3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
5-(4-chlorophenyl)-N-[2-(diethylamino)ethyl]-1,2,4-triazin-3-amine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3-{imidazo[1,2-a]pyridin-2-yl}propanamide
7-cyclopentyl-2-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
(3S,4R)-3-benzyl-4-methyl-1-(4-methyl-1H-imidazole-5-carbonyl)piperidin-4-ol
5-({2-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]ethyl}sulfanyl)-1H-1,2,3-triazole
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-(4-methylphenyl)ethan-1-one
3-[1-(3,6-dimethylpyrazin-2-yl)piperidin-3-yl]propanamide
1-[(4-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]-1,4-diazepan-5-one
2-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]-2-(3-hydroxyphenyl)acetic acid
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-{3-oxo-2-azaspiro[4.4]nonan-2-yl}acetamide
3-(4-chlorophenyl)-1-(furan-2-ylmethyl)piperidine
4-{[butyl(methyl)amino]methyl}-N-(dimethyl-1,2-oxazol-4-yl)benzamide
methyl 3-{[(2,2-dimethyloxan-4-yl)formamido]methyl}-5-(4-fluorobenzenesulfonamido)benzoate
(2S)-2-(morpholine-4-carbonyl)-N-[4-(1H-1,2,4-triazol-1-yl)phenyl]pyrrolidine-1-carboxamide
2-(5-acetylthiophen-3-yl)-N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)acetamide
3-methyl-3-[3-(oxolan-2-yl)propyl]-1-[4-(pyridin-3-yloxy)phenyl]urea
1-(1-methylpiperidin-4-yl)-4-(1H-pyrazole-4-carbonyl)-1,4-diazepan-6-ol
N-[2-({3-azaspiro[5.5]undecan-9-yl}amino)ethyl]pyridine-4-carboxamide
5-methyl-2-phenyl-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]furan-3-carboxamide
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N,5-dimethyl-2-phenyl-1H-imidazole-4-carboxamide
4-(2-methoxyethyl)-N-(4-oxo-4H-chromen-6-yl)piperazine-1-carboxamide
(4aR,7aS)-1-(2-methylpropyl)-4-(1H-pyrazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{4-[(pyrimidin-2-yl)amino]piperidin-1-yl}-N-(1,3-thiazol-2-yl)propanamide
1-[1-(morpholin-4-ylmethyl)cyclopentyl]-3-(1-oxo-1,3-dihydro-2-benzofuran-5-yl)urea
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl](methyl)[1-(pyridin-3-yl)propyl]amine
(4-{[5-(4-chlorophenoxy)-1,3-dimethyl-1H-pyrazol-4-yl]methyl}morpholin-2-yl)methanamine
1-(3-{[2-(2,3-dichlorophenyl)-1H-imidazol-1-yl]methyl}piperidin-1-yl)ethan-1-one
4-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-6-ethyl-2H-chromen-2-one