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N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]-1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-(propan-2-yl)piperazin-2-yl}ethan-1-ol
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-3-(furan-2-yl)propanamide
2-(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
[(3R,4R)-1-(5-chlorothiophene-2-carbonyl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
(1R,2R,6S,7S)-4-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
2-amino-4-(2-methoxypyrimidin-5-yl)-6-(4-methylphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-[4-(2-amino-6-methoxypyrimidin-4-yl)piperazin-1-yl]-1-(piperidin-1-yl)ethan-1-one
6-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-2-methyl-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
4-methoxy-N-{[1-(1,3-thiazole-4-carbonyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
2-methyl-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrido[2,3-d]pyrimidin-4-amine
2-(8-chloroquinoline-2-carbonyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decane
5-(2,4-difluorophenoxymethyl)-N-[(5,6-dimethylpyridin-3-yl)methyl]-1H-pyrazole-3-carboxamide
1-benzyl-N3-[(5-chlorothiophen-2-yl)methyl]-N5-cyclopropyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-methyl-5-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-1H-1,3-benzodiazole
5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-N-(pyridin-4-ylmethyl)pyrimidin-2-amine
1,3-dimethyl-4-[2-(trifluoromethyl)morpholin-4-yl]-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid
8-{5-[1-(morpholin-4-yl)propyl]-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl}quinoline
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-(pyridin-3-yl)pyrimidin-2-amine
2-(dimethylamino)-2-(2-fluorophenyl)-N-[2-methyl-2-(pyrrolidin-1-yl)propyl]acetamide
2-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrazine
N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamide
6-(6-methoxypyridin-3-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
N,5-dimethyl-N-[2-(pyridin-2-yl)ethyl]-1-benzofuran-2-carboxamide
(2S,4R)-4-amino-N-ethyl-1-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]pyrrolidine-2-carboxamide
{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}(2-methylpropyl)amine
methyl 6-({[(4-fluorophenyl)methyl](pyridin-4-ylmethyl)amino}methyl)pyridine-2-carboxylate
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-2-propyl-1,3-thiazole-4-carboxamide
1-cyclopropyl-N-[(5-methylthiophen-2-yl)methyl]-5-oxo-N-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
N-[3-(methylsulfanyl)propyl]-3-(piperidin-3-yl)benzamide
2-(adamantan-1-yl)-4-hydroxy-N-(1-hydroxypropan-2-yl)pyrimidine-5-carboxamide
5-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]pyrazine-2-carboxamide
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}acetamide
N-(furan-2-ylmethyl)-2-(2-oxopiperidin-1-yl)-N-(pyridin-2-ylmethyl)acetamide
3-(2H-1,3-benzodioxol-5-yl)-5-[4-(methylsulfanyl)butan-2-yl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N3-cyclohexyl-N3-methyl-N5-[(4-methylphenyl)methyl]-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-[3-(furan-2-yl)-5-(3-propyl-1H-pyrazol-4-yl)-1H-1,2,4-triazol-1-yl]acetic acid
(3aR,6aR)-2-(2-methoxyethyl)-5-[4-(methylsulfanyl)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
4-(6-{3-[1-(pyridin-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidin-4-yl)morpholine
2-(2,5-dioxoimidazolidin-4-yl)-N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]acetamide
1-(4-{[4-(2,3,4,9-tetrahydro-1H-carbazole-1-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
N-{1-[7-(cyclopent-1-ene-1-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-2-methylpropyl}pyridine-2-carboxamide
N-[3-(morpholin-4-yl)propyl]-2-[(prop-2-en-1-yl)amino]benzamide
2-methyl-6-{1-[2-(methylsulfanyl)benzoyl]piperidin-4-yl}pyrimidin-4-ol
2-(1H-indol-1-yl)-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-{[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]amino}hexanamide