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1-[(6-ethoxypyridin-3-yl)methyl]-4-{furo[3,2-c]pyridin-4-yl}piperazine
{2-[3-(naphthalene-1-carbonyl)piperidin-1-yl]-2-oxoethyl}urea
3-(3-hydroxyquinoxalin-2-yl)-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]propanamide
N-methyl-4-[4-(2-methylpropyl)phenyl]-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
2-[3-benzyl-1-(4-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N,N-diethylacetamide
(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-2-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-decahydroisoquinoline
(3R,4R)-N-(3-ethylphenyl)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidine-1-carboxamide
3-[(2-ethyl-2,5-dihydro-1H-pyrrol-1-yl)sulfonyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-5-(4-methylphenyl)-1H-pyrazole-3-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-(pyridin-4-yl)pyrimidin-2-amine
1,5,6-trimethyl-3-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-1,2-dihydropyridin-2-one
2-[4-(4-fluorophenyl)-4-hydroxypiperidin-1-yl]-N-[(2-methoxyphenyl)methyl]acetamide
1-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}azetidine
4-{1-cyclohexyl-5-[(methylsulfanyl)methyl]-1H-1,2,4-triazol-3-yl}pyridine
N-[(2-fluorophenyl)methyl]-3-[1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]propanamide
3-(3-chlorophenyl)-N-[2-(morpholin-4-yl)ethyl]-3-phenylpropanamide
2-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-2,8-diazaspiro[4.5]decane
N-{3-[2-(2-hydroxyethyl)-3-oxopiperazine-1-carbonyl]-2-methylphenyl}furan-2-carboxamide
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-3-(1H-pyrazol-1-yl)butan-1-one
N-(butan-2-yl)-4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}benzamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[2-hydroxy-2-(1-methyl-1H-imidazol-2-yl)ethyl]acetamide
N-{2-[4-(3-methyl-1H-1,2,4-triazol-5-yl)phenoxy]ethyl}acetamide
7-(2-hydroxybenzoyl)-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(4-methoxyphenyl)-4-{1-[4-(methylsulfanyl)benzoyl]piperidin-3-yl}piperazine
(1S,5R)-6-(2-methoxyethyl)-3-[(2-phenylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-[(3-methylfuran-2-yl)formamido]-N-(naphthalen-1-yl)propanamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-[(1-methyl-1H-imidazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(pyrazin-2-yl)propan-1-one
6-(2,5-dimethylfuran-3-yl)-8-oxo-7-(prop-2-en-1-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-({1-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-4-hydroxyazepan-4-yl}methyl)-3,3-dimethylurea
(2R,3R)-3-[4-(3-fluorophenyl)-1H-1,2,3-triazol-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-3-yl)benzoic acid
(3S)-3-{[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]amino}azepan-2-one
1-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}azetidin-3-ol
6-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
1-cyclopropyl-3-{4-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-1-(pyridin-4-ylmethyl)urea
1-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propane-1,2-dione
3-cyclohexyl-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
5-({4-[4-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)quinoline
1-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-2-(4-methyl-1H-pyrazol-1-yl)propan-1-one
[(3R,5R)-5-[(dimethylamino)methyl]-1-[2-(1H-imidazol-2-yl)benzoyl]piperidin-3-yl]methanol
1-methyl-4-{6-methylimidazo[2,1-b][1,3]thiazol-5-yl}-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{1-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopentanecarboxamide
7-(cyclopropylmethyl)-2-[3-(1H-imidazol-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
7-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-amino-4-(2-chloro-6-fluorophenyl)-6-(pyridin-2-yl)pyridine-3-carbonitrile
5-{[(3-methyl-1-benzofuran-2-yl)methyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
3-[(3S,7S,8aS)-1,4-dioxo-3-propyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-2-methylphenyl)urea
4-{[3-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-N-methylbenzene-1-sulfonamide
4-(1-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidin-3-yl)morpholine