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5-(2-chlorophenyl)-N-[cyclopropyl(1-methyl-1H-1,2,4-triazol-5-yl)methyl]furan-2-carboxamide
4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-N-(1,2,2,6,6-pentamethylpiperidin-4-yl)pyrimidin-2-amine
2-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-5-phenyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-2-one
N-ethyl-N-(pyridin-4-ylmethyl)oxane-2-carboxamide
(3R,4S)-1-[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazole-4-carbonyl]-4-phenylpyrrolidin-3-amine
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-{1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]azetidin-3-yl}pyridine
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
3-chloro-4-fluoro-N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-benzothiophene-2-carboxamide
1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-phenoxypropan-1-one
N-[2-(3-chlorophenoxy)ethyl]-N-ethyloxolane-3-carboxamide
(2R,4S)-4-hydroxy-1-(thiophene-2-carbonyl)piperidine-2-carboxylic acid
N-({5-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(6-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(1-benzylpiperidin-4-yl)-N-methyl-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
methyl 3-[(3S,4R)-4-(dimethylamino)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-3-yl]propanoate
7-(1-methyl-1H-pyrrole-2-carbonyl)-N-(oxan-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-4-(naphthalen-1-yl)-1H-1,2,3-triazole
5-ethyl-N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-1,3,4-oxadiazol-2-amine
methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]{[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}amine
N-[3-(5-chloro-1H-1,3-benzodiazol-2-yl)propyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
1-{2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
3-cyano-N-[2-(dimethylamino)ethyl]-5-fluoro-N-(oxolan-2-ylmethyl)benzamide
4-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-N-methyl-4-oxobutanamide
(3S,4R)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
1-{4-[3-(4-ethylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
1-(2-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-2-yl}ethyl)-4-methylpiperazine
N-(1-{5-[(cyclohexylmethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-3-fluorobenzene-1-sulfonamide
2-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidine-1-carbonyl]pyridin-3-ol
5-oxo-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-1-(prop-2-en-1-yl)pyrrolidine-3-carboxamide
4-(furan-2-ylmethyl)-3-[1-(morpholin-4-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1,3-oxazole-4-carboxamide
N-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-N-methyl-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
5-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-N-[(4-fluorophenyl)methyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(pyridin-3-yl)-4-[2-(pyridin-4-yl)-1H-imidazol-1-yl]benzamide
2-({3-[(dicyclopropylmethyl)(methyl)carbamoyl]phenyl}amino)acetic acid
5-oxo-1-(propan-2-yl)-N-[2-(1,3-thiazol-2-yl)ethyl]pyrrolidine-3-carboxamide
3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}-3-({[2-(1H-1,2,3-triazol-1-yl)ethyl]amino}methyl)piperidin-2-one
6-ethyl-3-[2-(piperazin-1-yl)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-6-ethyl-2-methylquinoline-4-carboxamide
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-(dimethylamino)-2-(2-methylphenyl)ethan-1-one
N-[(3-methoxyphenyl)methyl]-3-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}propanamide
2-ethyl-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)pyrimidine-5-carboxamide
2-(3,4-difluorophenyl)-5-[(2,3,4-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
6-methyl-N4-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-5-(prop-2-en-1-yl)pyrimidine-2,4-diamine
N3-methyl-4-oxo-1-(2-phenylethyl)-N5-[1-(thiophen-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-(3-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}phenyl)ethan-1-one
N,N-diethyl-1-{1-[(5-methylthiophen-2-yl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
N-(3,4-dimethoxyphenyl)-2,7-diazaspiro[4.5]decane-7-carboxamide