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7-(3-chlorophenyl)-4-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(furan-2-yl)-2-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethane-1,2-dione
5-phenyl-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-2-(1H-pyrazol-1-yl)butanamide
ethyl 5-[(4-carbamoylpiperidin-1-yl)methyl]-1-(4-fluorophenyl)-1H-pyrazole-4-carboxylate
butyl (1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
4-({2-[1-(1H-pyrazole-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
4-(4-benzyl-1H-pyrazol-5-yl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
1-(2-chloro-6-methylphenyl)-3-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]urea
2-[(4aR,7aS)-4-[(3,4-dimethylphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
2-(cyclopropylmethyl)-9-[(3-fluoro-5-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(1R,5R)-3-cyclobutanecarbonyl-6-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-(3-{[(8-methoxy-4-methylquinolin-2-yl)amino]methyl}pyridin-2-yl)piperidin-3-ol
(4aS,8aR)-6-(1H-imidazole-2-carbonyl)-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
(3aR,6aR)-2-[(2-phenylethyl)carbamoyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidine-1-carboxamide
2-amino-7-(2,3,4,9-tetrahydro-1H-carbazole-6-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-(3-hydroxy-3-methylbutyl)-N-[2-(1H-imidazol-4-yl)ethyl]benzamide
1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
5-(3-acetylphenoxymethyl)-N-(pyrrolidin-3-ylmethyl)-1,2-oxazole-3-carboxamide
4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-7-hydroxy-6-methyl-1,2,3,4-tetrahydroquinolin-2-one
4-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-2-ethylmorpholine
3-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
2-(4-{1-[2-(phenylsulfanyl)ethyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)ethan-1-ol
N-{2-[(2S)-pyrrolidin-2-yl]ethyl}-2-(4H-1,2,4-triazol-4-yl)benzamide
8-[5-(3-methoxyphenyl)furan-2-carbonyl]-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
5-methyl-4-[2-(pyridin-4-yl)-1H-imidazol-1-yl]-2,1,3-benzothiadiazole
2,6-dimethyl-4-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]quinoline
1-methyl-2-oxo-N-[1-(thiophen-3-yl)ethyl]-1,2-dihydroquinoline-4-carboxamide
N-cyclopropyl-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
3-(1-cyclopentyl-1H-pyrazol-5-yl)-1-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}urea
1-[(3,5-dimethoxyphenyl)methyl]-3-[2-(methylsulfanyl)benzoyl]piperidine
5-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-N-phenyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
2-(4-fluorophenyl)-4-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)morpholine
N-ethyl-N-(pyridin-4-ylmethyl)-1-(quinoline-8-sulfonyl)piperidin-3-amine
5-[4-(4-methoxyphenyl)butanoyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-fluoro-N-[(3S)-2-oxoazepan-3-yl]-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)benzamide
{[2-(methoxymethyl)pyrimidin-5-yl]methyl}({[4-(methylsulfanyl)phenyl]methyl})propylamine
8-(2-methoxypyridin-3-yl)-2-(pyrrolidin-1-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
N-methyl-N-(2-methylpropyl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
N-methyl-2-[({2-[(naphthalen-1-yl)amino]-1,3-thiazol-5-yl}methyl)amino]ethane-1-sulfonamide
N-{1-[1-(2-aminopyrimidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-methoxybenzamide
N-(1-{1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methylthiophene-3-carboxamide
[3-(3-{2-azaspiro[4.4]nonan-2-ylmethyl}phenoxy)propyl]dimethylamine
5-[1-(3-ethyl-1H-indole-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
5-[2-(ethylamino)ethyl]-1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-one
2-{5-[6-amino-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-[1-(pyridin-2-yl)propyl]acetamide