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3-(2-{3-[(naphthalen-1-ylformamido)methyl]piperidin-1-yl}-2-oxoethyl)-1,2,3-oxadiazol-3-ium-5-olate
4-[2-(2,4,7-trimethyl-1H-indol-3-yl)acetyl]piperazin-2-one
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]piperidine-3-carboxamide
4-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-2-(4-fluorophenyl)morpholine
methyl (2S)-1-[2-(4-{4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-1-yl}phenyl)acetyl]pyrrolidine-2-carboxylate
(3S,9aR)-8-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-methyl-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]pyrazin-2-ol
2-(hydroxymethyl)-N-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}piperidine-1-carboxamide
3-(hydroxymethyl)-1-({2-[3-(morpholin-4-yl)propoxy]phenyl}methyl)piperidin-3-ol
5-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}pyrazin-2-ol
1-methyl-2-(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-4-yl)-1H-1,3-benzodiazole
3-{1-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-3-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-[(3S,5S)-1-[(2,5-dimethylphenyl)methyl]-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
(1S,5R)-3-(2-amino-5,6-dimethylpyrimidin-4-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{1-[1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(3-fluorophenyl)urea
2-{[1-(2,3-dihydro-1H-inden-5-yl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]methoxy}acetamide
4-[2-amino-3-cyano-6-(2,3-dihydro-1,4-benzodioxin-6-yl)pyridin-4-yl]benzamide
4-(3-{3-[3-(furan-3-yl)phenyl]-1H-pyrazol-1-yl}propyl)morpholine
2-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-[9-(5-methylthiophene-2-carbonyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
2-{[4-(5-fluoropyrimidin-2-yl)piperazin-1-yl]methyl}quinolin-4-ol
(2S,4S)-4-amino-1-{[3-(difluoromethoxy)phenyl]methyl}-N,N-diethylpyrrolidine-2-carboxamide
5-methyl-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-6-[(2-methylpyridin-3-yl)oxy]pyrimidine
3-(carbamoylmethoxy)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
1-[2-(2-ethylphenoxy)ethyl]-3-methoxy-1,2-dihydropyridin-2-one
2-(3-fluorophenyl)-N-(4-{4-[(thiophen-3-ylmethyl)amino]piperidin-1-yl}phenyl)acetamide
3-{[(4-fluorophenyl)methyl]sulfanyl}-N-[(4-hydroxy-3-methoxyphenyl)methyl]propanamide
1-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-3,3-dimethylurea
5-{3-[4-(benzyloxy)piperidin-1-yl]-3-oxopropyl}-5-[(4-methylphenyl)methyl]pyrrolidin-2-one
6-oxo-N-[3-(pyridin-3-yl)propyl]-1,4,5,6-tetrahydropyridazine-3-carboxamide
5-chloro-4-[5-(methanesulfonylmethyl)pyridin-2-yl]-2-methoxypyridine
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(3-methoxybenzoyl)piperazine
1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
2-({3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}amino)propan-1-ol
5-ethyl-N-[4-(pyrrolidin-1-yl)butyl]pyrazolo[1,5-a]pyrimidin-7-amine
6-acetyl-2-amino-4-(2-chloro-4-hydroxy-5-methoxyphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-(3-chloro-4-methoxyphenyl)-N-[2-(1H-imidazol-1-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-4,6-dimethyl-2-oxo-2H-pyran-5-carboxamide
3-hydroxy-3-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}-1-[(3-methylphenyl)methyl]piperidin-2-one
methyl({[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl})[2-(pyrrolidin-1-yl)ethyl]amine
2-cyclopentyl-1-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
N-benzyl-6,6-dimethyl-5-oxo-N-(1,3-thiazol-2-ylmethyl)thiomorpholine-3-carboxamide
1-cyclopentyl-3-(2-fluorophenyl)-3-{2-oxo-2-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]ethyl}pyrrolidine-2,5-dione
4-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propanoyl]-1-(2-methylphenyl)piperazin-2-one
7-(1,3-benzothiazol-2-yl)-4-(4-methyl-1H-imidazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N,1-dimethyl-3-(2-methylpropyl)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1H-pyrazole-5-carboxamide
7-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-N,N-dimethyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-methyl-N-[7-oxo-5-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]butanamide
3-({4-[1-ethyl-3-(hydroxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-6-methylpyrimidin-2-yl}amino)phenol