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4-oxo-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
3-(3-methoxyphenoxy)-1-(3,3,3-trifluoro-2-methylpropyl)azetidine
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(2,2-dimethyloxan-4-yl)-N-ethylbenzamide
(1R,2R,6S,7S)-4-{6-cyclopropyl-3-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-10-oxa-4-azatricyclo[5.2.1.02,6]decane
2-(dimethylamino)-2-(3-fluorophenyl)-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)acetamide
4-[(4-fluoro-2-methylphenyl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
4-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
1-{2-amino-4-[(2-hydroxyethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-(pyridin-3-yloxy)ethan-1-one
3-[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)pyrrolidin-2-yl]-5-(propan-2-yl)-1,2-oxazole
1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
dimethyl(2-{1-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]piperidin-2-yl}ethyl)amine
N-(1,4-dioxan-2-ylmethyl)-4-(piperidin-1-yl)benzamide
(1S,4S)-2-[5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-2-azabicyclo[2.2.1]heptane
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(2-methoxyphenyl)acetamide
3-(5-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
(3aS,7aR)-5-methyl-2-(2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[(3S)-2-oxoazepan-3-yl]benzamide
1-(4-hydroxyphenyl)-2-[methyl(quinolin-4-ylmethyl)amino]ethan-1-one
2-(4,6-dimethyl-1-benzofuran-3-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-(2-methoxyethyl)-5-(4-methoxyphenyl)-N-(1-methylpiperidin-4-yl)furan-2-carboxamide
1-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
2-(5-{2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]ethyl}-3-(3-methylphenyl)-1H-1,2,4-triazol-1-yl)ethan-1-ol
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-ethyl-4-methyl-N-(propan-2-yl)-1,3-oxazole-5-carboxamide
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-methyl-4-{1-[1-(pyridin-4-yl)piperidin-4-yl]ethyl}piperazine
2-{methyl[5-({methyl[1-(pyridin-4-yl)ethyl]amino}methyl)pyrimidin-2-yl]amino}acetic acid
[2-ethoxy-5-({methyl[2-(methylamino)ethyl]amino}methyl)phenyl]methanol
3-(propan-2-yl)-N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-1H-pyrazole-5-carboxamide
1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carboxamide
6-({4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}methyl)-N-[(1-hydroxycyclohexyl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]phenol
6-[(diethylamino)methyl]-N-methyl-N-(thiophen-3-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-[2-(1H-pyrazol-1-yl)ethyl]-1-(1H-1,2,4-triazole-5-carbonyl)piperidine
5-{[3-(3-methylbutoxy)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-chloro-2-{[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]methyl}phenol
N-(4-acetamidophenyl)-4-[(2-ethyl-2,5-dihydro-1H-pyrrol-1-yl)methyl]benzamide
6-{1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]piperidin-3-yl}-3,4-dihydropyrimidin-4-one
2-(4-chloro-1H-pyrazol-1-yl)-1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]propan-1-one
7-methyl-3-{2-[1-(propan-2-yl)piperidin-2-yl]ethyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
6-chloro-4-[4-(1H-imidazol-2-yl)piperidin-1-yl]-8-methylquinoline
N-cyclohexyl-N-methyl-4-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
N,N-bis(furan-2-ylmethyl)-9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
4-({[2-(4-methoxyphenyl)ethyl]carbamoyl}methyl)piperazine-1-carboxamide
4-({5-[1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
(2S,4R)-N-methyl-4-[(naphthalen-2-ylmethyl)amino]-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-[(5-methylfuran-2-yl)methyl]-3-[1-(quinoxaline-5-carbonyl)piperidin-3-yl]propanamide
4-(hydroxymethyl)-1-{[1-(3-methylbutyl)-1H-1,3-benzodiazol-2-yl]methyl}azepan-4-ol
1-[4-({4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}methyl)thiophen-2-yl]ethan-1-one
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine