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N-methyl-3-(6-oxo-1,6-dihydropyridazin-3-yl)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]propanamide
2-[2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidin-4-yl]pyridine-4-carboxylic acid
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(1-methyl-1H-imidazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-methyl-5-(pyrrolidine-1-sulfonyl)-2-(trimethyl-1H-pyrazol-4-yl)-1H-1,3-benzodiazole
(2S,4R)-4-amino-N-methyl-1-(1-propyl-1H-pyrazole-5-carbonyl)pyrrolidine-2-carboxamide
4-methoxy-2-{[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}phenol
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]pyrimidine
5-{[2-(ethylsulfanyl)-1,3-thiazol-4-yl]methyl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-(3-methyl-4-{[(2S)-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]methyl}-1H-pyrazol-1-yl)ethan-1-ol
8-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(4-methyl-1H-imidazole-2-carbonyl)piperidine
5-methoxy-N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)furan-2-carboxamide
3-methyl-1-(5-{[methyl(2-phenylethyl)amino]methyl}-1,2-oxazole-3-carbonyl)piperidin-3-ol
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,2-dimethyl-1H-pyrrole-3-carboxamide
(1H-imidazol-2-ylmethyl)(methyl){[5-(oxan-2-yl)furan-2-yl]methyl}amine
4-[(4-fluorophenyl)methyl]-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
5-{1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1H-1,2,3-triazol-4-yl}-2-methoxypyridine
1-[3-(2,4-dimethoxybenzoyl)piperidine-1-carbonyl]cyclopropan-1-amine
1-{[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-5-methyl-1-phenylpiperazin-2-one
1-(morpholin-4-yl)-2-[4-({[1-(1H-pyrazol-1-yl)propan-2-yl]amino}methyl)phenoxy]ethan-1-one
2-ethyl-N,4-dimethyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1,3-oxazole-5-carboxamide
7-[(3,5-difluoro-4-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
2-{2-hydroxy-2-[2-(trifluoromethyl)phenyl]ethyl}-2,9-diazaspiro[5.5]undecan-3-one
1-(2-methoxyethyl)-3-(naphthalen-1-ylmethyl)-8-[4-(1H-pyrazol-1-yl)butan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-5,6-dimethylpyrimidin-4-amine
5-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonane-7-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
2,5-dimethyl-4-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine
2-(5-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-N-methyl-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
N-[4-(1H-pyrazol-1-yl)phenyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carboxamide
5-oxo-1-(prop-2-en-1-yl)-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]pyrrolidine-3-carboxamide
1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-fluoro-2-phenylethan-1-one
4-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
N-[1-(3-methylphenyl)piperidin-4-yl]-6-oxo-1,6-dihydropyridine-2-carboxamide
2-(4-methoxy-3,5-dimethylphenyl)-2-[methyl(2-methylprop-2-en-1-yl)amino]acetic acid
1-methyl-N-[3-(3-methylpiperidin-1-yl)propyl]-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-propylcyclopropan-1-amine
1-(6-aminopyrimidin-4-yl)-3-[(2,4-difluorophenyl)methyl]piperidine-3-carboxylic acid
4-[2-(4-benzyl-3-butyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetyl]piperazin-2-one
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-5,6,7-trimethoxy-1,2-dihydroquinolin-2-one
3-(2-{2-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1H-imidazol-1-yl}ethyl)-5-methyl-1,2,4-oxadiazole
8-(3-chloro-4-methoxybenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-cyclohexyl-3-{[2-(ethylamino)pyrimidin-5-yl]formamido}propanamide
2-{2-[2-amino-3-cyano-5-ethyl-6-(propan-2-yl)pyridin-4-yl]phenoxy}-N,N-dimethylacetamide
9-[5-(2-chlorophenyl)furan-2-carbonyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
4-({2-amino-4-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}methyl)benzoic acid
8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-[(3-fluoro-4-methylphenyl)methyl]propanamide
(3aS,6aS)-2-cyclohexyl-5-(1,3-thiazol-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid