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1-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
1-{[1-(1-benzoxepine-4-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
1-{2-[3-(4-methylphenoxymethyl)piperidin-1-yl]-2-oxoethyl}azepan-2-one
methyl[(2-methyl-1,3-thiazol-4-yl)methyl][(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amine
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methyloxolan-3-amine
N-methyl-5-propyl-N-(pyrazin-2-ylmethyl)-1,3,4-oxadiazole-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-{[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
(2S,4R)-4-amino-1-[3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[1-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-3-phenoxypropanamide
(3R,4R)-1-[1-(benzenesulfonyl)cyclopropanecarbonyl]-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
(3R,4R)-4-(azepan-1-yl)-1-[(5-chloro-2,3-dimethoxyphenyl)methyl]piperidin-3-ol
3-(3-fluorophenyl)-N-[(4-methanesulfonylmorpholin-2-yl)methyl]-1H-pyrazole-4-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}acetamide
2-[4-(morpholin-4-ylmethyl)phenyl]-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
5-fluoro-2-(1-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
(2R,6R)-11-methoxy-4-[2-(thiophen-3-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
9-methoxy-7-(3-methoxyphenyl)-4-(thiophen-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1R,3S,5S)-8-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-8-azabicyclo[3.2.1]octan-3-ol
2-(2-phenyl-1,3-thiazol-4-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}acetamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(oxane-4-carbonyl)pyrrolidine-3-carboxylic acid
4-methoxy-N-methyl-3-({[1-(pyrimidin-2-yl)piperidin-3-yl]carbamoyl}amino)benzamide
2-methyl-7-[(1-propyl-1H-imidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decane
2-{5-[(3-cyclohexylpyrrolidin-1-yl)methyl]-1,2,4-oxadiazol-3-yl}pyridine
1-(4,7-dimethylquinazolin-2-yl)-N-(3-hydroxyadamantan-1-yl)piperidine-3-carboxamide
(3R,4R)-1-(5-methoxyfuran-2-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
1-{2-[methyl({[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl})amino]pyrimidin-4-yl}pyrrolidin-3-ol
N-(3-hydroxy-3-phenylpropyl)-N,1-dimethyl-1H-indole-4-carboxamide
6-methyl-3-(2-methylpiperidine-1-carbonyl)-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridin-4-one
1-[5-(methoxymethyl)furan-2-carbonyl]-3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
5-(2-chlorophenyl)-N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]furan-2-carboxamide
4-{4-[(3-ethoxy-4-methoxyphenyl)methyl]piperazin-1-yl}-2-[2-(2-fluorophenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
3-[(2,6-dimethoxyphenyl)methyl]-8-methoxy-3,4-dihydroquinazolin-4-one
4-(2,1,3-benzoxadiazol-5-yl)-1-benzyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(2-methylpropyl)pyrrolidin-3-yl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
(2E)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-2-methyl-N-(2-methylpropyl)but-2-enamide
3-methoxy-1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]pyrrolidine
4-[4-(piperidine-1-sulfonyl)-1,4-diazepane-1-carbonyl]pyridin-3-ol
3-[5-(6-aminopyridine-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-N-cyclopropylpropanamide
N-(5-methyl-1,2-oxazol-3-yl)-2-(2-methylpyrimidine-5-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
3-{1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
9-(5-methylpyridine-2-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{4-[3-(benzyloxy)piperidin-1-yl]piperidin-1-yl}-7-methanesulfonyl-4-methylquinazoline
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-[2-(pyrazin-2-yl)acetyl]pyrrolidin-3-yl]urea
2-(2,3,4,9-tetrahydro-1H-carbazole-6-carbonyl)-1,2,3,4-tetrahydroisoquinolin-4-ol
2-chloro-N-(2-{[2-(dimethylamino)pyridin-3-yl]formamido}ethyl)benzamide
5-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidine-1-carbonyl}-2-methyl-1,4-dihydropyridin-4-one
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)-2-[3-(trifluoromethyl)phenyl]acetamide
[(3R,4R)-4-(pyrrolidin-1-ylmethyl)-1-(1,3,4-thiadiazol-2-yl)pyrrolidin-3-yl]methanol
N-(2-methanesulfonylethyl)-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide